Agonists |
Dopamine | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 474 | 25 | 19 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 710 | 29 | 24 |
Freedman et al. (1994)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 710 | 15 | 46 |
Kula et al. (1994)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 540 | 23 | 23 |
Sautel et al. (1995a)
|
| [125I]NCQ-298 | hD2L/HEK 293 | rD3/HEK 293 | 1908 | 44 | 43 |
Burris et al. (1995) |
| [125I]7-OH-PIPAT | hD2L/HEK 293 | rD3/HEK 293 | 5.8 | 5.6 | 1.0 |
Burris et al. (1995)
|
| [3H]N-0437 | hD2L/CHO-K1 | hD3/CHO-K1 | 31 | 11 | 2.8 |
Pugsley et al. (1995)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 8.5 | 4.8 | 1.8 |
Flietstra and Levant (1996)
|
|
Bromocriptine | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 5.3 | 7.4 | 0.72 |
Sokoloff et al. (1990)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 33 | 49 | 0.67 |
Levant and DeSouza (1993)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 0.62 | 2.1 | 0.30 |
Freedman et al. (1994b)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 0.067 | 0.20 | 0.34 |
Kula et al. (1994)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 5.3 | 7.4 | 0.72 |
Sautel et al. (1995a)
|
| [3H]pramipexole | hD2L/HEK 293 | hD3/DHO dhfr- | 2.5 | 12.2 | 0.21 |
Mierau et al. (1995)
|
|
Apomorphine | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 24 | 20 | 1.2 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 63 | 73 | 0.86 |
Sokoloff et al. (1992)
|
| [3H]spiperone | hD2/CHO-K1 | hD3/CHO-K1 | 24 | 9.3 | 2.6 |
MacKenzie et al. (1994)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 30 | 16 | 1.9 |
Freedman et al. (1994)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 34 | 23 | 1.5 |
Kula et al. (1994)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 63 | 73 | 0.86 |
Sautel et al. (1995a)
|
| [125I]NCQ-298 | hD2L/HEK 293 | rD3/HEK 293 | 168 | 31 | 5.4 |
Burris et al. (1995) |
| [125I]7-OH-PIPAT | hD2L/HEK 293 | rD3/HEK 293 | 4.9 | 14 | 0.35 |
Burris et al. (1995)
|
| [3H]N-0437 | hD2L/CHO-K1 | hD3/CHO-K1 | 2.9 | 8.9 | 0.33 |
Pugsley et al. (1995)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 47 | 23 | 2.0 |
Millan et al. (1995b)
|
|
Quinpirole | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 576 | 5.1 | 113 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 1402 | 39 | 36 |
Sokoloff et al. (1992)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 3.7 | 3.6 | 1.0 |
Levant and De Souza (1993)
|
| [3H]spiperone | hD2/CHO-K1 | hD3/CHO-K1 | 193 | 5.3 | 36 |
MacKenzie et al. (1994)
|
| [3H]spiperone | rD2L/CCL1.3 | hD3/CCL1.3 | 15 | 19 | 0.80 |
Tang et al. (1994a)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 1920 | 32 | 60 |
Kula et al. (1994)
|
| [125I]NCQ-298 | hD2L/HEK 293 | rD3/HEK 293 | 1065 | 8.0 | 133 |
Burris et al. (1995) |
| [125I]7-OH-PIPAT | hDSL/HEK 293 | rD3/HEK 293 | 6.4 | 1.7 | 3.8 |
Burris et al. (1995)
|
| [125I]iodosulpiride1-a
| rStriatum | rCerebellar lob.X | 1571-b
| 281-b
| 5.6 |
Levant et al. (1995) |
| [3H]pramipexole | hD2L/HEK 293 | hD3/DHO dhfr- | 1.8 | 0.96 | 1.9 |
Mierau et al. (1995)
|
| [3H]N-0437 | hD2L/CHO-K1 | hD3/CHO-K1 | 82 | 9.3 | 8.8 |
Pugsley et al. (1995)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 911 | 43 | 21 |
Millan et al. (1995)
|
|
Quinelorane | [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 341 | 3.6 | 95 |
Sokoloff et al. (1992)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 265 | 6.1 | 43 |
Millan et al. (1995)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 5.7 | 3.4 | 1.7 |
Fliestra and Levant (1996)
|
|
7-OH-DPAT | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 61 | 0.78 | 78 |
Lévesque et al. (1992)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 30 | 5.8 | 5.2 |
Levant and De Souza (1993)
|
| [3H]spiperone | hD2/CHO-K1 | hD3/CHO-K1 | 156 | 1.6 | 98 |
MacKenzie et al. (1994)
|
| [3H]spiperone | hD2/CCL1.3 | hD3/CCL1.3 | 223 | 7.1 | 31 |
MacKenzie et al. (1994)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 60 | 1.6 | 38 |
Freedman et al. (1994)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 160 | 3.8 | 42 |
Kula et al. (1994)
|
| [125I]7-OH-PIPAT | hD2/sf9 | hD3/sf9 | 142 | 2.9 | 49 |
Chumpradit et al. (1994)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 103 | 2.1 | 49 |
Sautel et al. (1995a)
|
| [125I]NCQ-298 | hD2L/HEK 293 | rD3/HEK 293 | 165 | 1.2 | 138 |
Burris et al. (1995) |
| [125I]7-OH-PIPAT | hD2L/HEK 293 | rD3/HEK 293 | 2.6 | 0.4 | 6.5 |
Burris et al. (1995)
|
| [125I]iodosulpiride1-a
| rStriatum | rCerebellar lob.X | 991-b
| 4.21-b
| 24 |
Levant et al. (1995)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 103 | 2.2 | 47 |
Millan et al. (1995)
|
|
(−)-N-prophynor- | [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 0.12 | 0.21 | 0.57 |
Freedman et al. (1994)
|
apomorphine | [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 3.4 | 0.27 | 13 |
Kula et al. (1994)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 2.9 | 0.36 | 8.1 |
Sautel et al. (1995a)
|
Pramipexole | [125I]iodosulpiride | hD2/CHO | hD3/CHO | 790 | 4.1 | 193 |
Sautel et al. (1995a)
|
| [3H]pramipexole | hD2L/HEK 293 | hD3/CHO dhfr- | 3.9 | 0.5 | 7.8 |
Mierau et al. (1995) |
|
PD 128907 | [3H]N-0437 | hD2L/CHO-K1 | hD3/CHO-K1 | 42 | 2.3 | 18 |
Pugsley et al. (1995)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 389 | 1.8 | 216 |
Sautel et al. (1995a)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 109 | 18 | 6.1 |
Flietstra and Levant (1996)
|
|
7-trans-OH- | [125I]7-OH-PIPAT | hD2/sf9 | hD3/sf9 | 265 | 1.9 | 143 |
Chumpradit et al. (1994)
|
PIPAT | [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 20 | 47 | 0.43 |
Flietstra and Levant (1996)
|
Antagonists |
Domperidone | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 0.30 | 9.5 | 0.03 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 1.3 | 7.5 | 0.17 |
Sokoloff et al. (1992)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 0.58 | 2.9 | 0.20 |
Freedman et al. (1994)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 0.5 | 3.5 | 0.14 |
Millan et al. (1995)
|
| [125I]iodosulpiride1-a
| rStriatum | rCerebellar lob.X | 4.51-b
| 831-b
| 0.05 |
Levant et al. (1995)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 3.4 | 125 | 0.027 |
Flietstra and Levant (1996)
|
|
Haloperidol | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 0.45 | 9.8 | 0.05 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 0.6 | 2.9 | 0.21 |
Sokoloff et al. (1992)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 17 | 1020 | 0.017 |
Levant and De Souza (1993)
|
| [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 0.67 | 2.74 | 0.24 |
Malmberg et al. (1993)
|
| [3H]spiperone | hD2/CHO-K1 | hD3/CHO-K1 | 0.3 | 1.0 | 0.30 |
MacKenzie et al. (1994)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 2.6 | 1.5 | 1.73 |
Freedman et al. (1994)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 0.90 | 1.91 | 0.47 |
Kula et al. (1994)
|
| [125I]iodosulpiride1-a
| rStriatum | rCerebellar lob.X | 6.31-b
| 231-b
| 0.27 |
Levant et al. (1995) |
| [3H]pramipexole | hD2L/HEK 293 | hD3/DHO dhfr- | 0.17 | 2.9 | 0.059 |
Mierau et al. (1995) |
| [3H]N-0437 | hD2L/CHO-K1 | hD3/CHO-K1 | 0.27 | 2.8 | 0.10 |
Pugsley et al. (1995)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 0.45 | 2.4 | 0.19 |
Millan et al. (1995)
|
|
Spiperone | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 0.069 | 0.61 | 0.11 |
Sokoloff et al. (1990)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 0.35 | 28 | 0.013 |
Levant and De Souza (1993)
|
| [3H]spiperone | hD2/CHO-K1 | hD3/CHO-K1 | 0.2 | 0.3 | 0.67 |
MacKenzie et al. (1994)
|
| [3H]spiperone | hD2/CCL1.3 | hD3/CCL1.3 | 0.37 | 0.32 | 1.16 |
MacKenzie et al. (1994) Tang et al. (1994)
|
| [3H]spiperone | rD2L/MN9D | hD3/MN9D | 0.28 | 0.71 | 0.39 |
Tang et al. (1994)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 0.017 | 0.030 | 0.57 |
Kula et al. (1994)
|
| [125I]iodosulpiride1-a
| rStriatum | rCerebellar lob.X | 2.11-b
| 3.41-b
| 0.62 |
Levant et al. (1995)
|
| [3H]N-0437 | hD2L/CHO-K1 | hD3/CHO-K1 | 0.10 | 0.4 | 0.25 |
Pugsley et al. (1995)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 0.06 | 0.25 | 0.24 |
Millan et al. (1995)
|
|
Clozapine | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 56 | 180 | 0.31 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 69 | 479 | 0.14 |
Sokoloff et al. (1992)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 1575 | 9633 | 0.16 |
Levant and De Souza (1993)
|
| [3H]raclopride | hD2L/Ltk- | hD3Ltk- | 60 | 83 | 0.72 |
Malmberg et al. (1993)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 38 | 88 | 0.43 |
Freedman et al. (1994)
|
| [3H]spiperone | hD2/CHO-K1 | hD3/CHO-K1 | 17 | 264 | 0.064 |
MacKenzie et al. (1994)
|
| [3H]spiperone | hD2/CCL1.3 | hD3/CCL1.3 | 143 | 620 | 0.23 |
MacKenzie et al. (1994) Tang et al. (1994)
|
| [3H]siperone | rD2L/MN9D | hD3/MN9D | 170 | 480 | 0.35 |
Tang et al. (1994)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 125 | 158 | 0.79 |
Kula et al. (1994)
|
|
(−)-Sulpiride | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 9.2 | 25 | 0.37 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 10 | 20 | 0.50 |
Sokoloff et al. (1992)
|
| [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 7.4 | 8.0 | 0.93 |
Malmberg et al. (1993)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 6.0 | 8.0 | 0.75 |
Freedman et al. (1994)
|
| [3H]spiperone | hD2/CCL1.3 | hD3/CCL1.3 | 72 | 570 | 0.13 |
MacKenzie et al. (1994)
|
| [3H]spiperone | rD2L/MN9D | hD3/MN9D | 57 | 207 | 0.28 |
Tang et al. (1994)
|
| [125I]NCQ-298 | hD2L/HEK 293 | rD3/HEK 293 | 12 | 14 | 0.86 |
Burris et al. (1995) |
| [125I]7-OH-PIPAT | hD2L/HEK 293 | rD3/HEK 293 | 60 | 142 | 0.42 |
Burris et al. (1995)
|
| [125I]iodosulpiride1-a
| rStriatum | rCerebellar lob.X | 111-b
| 6.31-b
| 1.8 |
Levant et al. (1995)
|
Amisulpiride | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 1.7 | 3.8 | 0.45 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 1.3 | 2.4 | 0.54 |
Sokoloff et al. (1992)
|
| [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 0.97 | 3.0 | 0.32 |
Malmberg et al. (1993)
|
|
Chlorpromazine | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 2.8 | 6.1 | 0.46 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 2.3 | 5.9 | 0.39 |
Sokoloff et al. (1992)
|
| [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 1.14 | 1.16 | 0.98 |
Malmberg et al. (1993)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 8.0 | 3.0 | 2.7 |
Freedman et al. (1994)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 29 | 114 | 0.25 |
Flietstra and Levant (1996)
|
|
Raclopride | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 1.8 | 3.5 | 0.51 |
Sokoloff et al. (1990)
|
| [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 2.3 | 1.8 | 1.28 |
Malmberg et al. (1993)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 1.1 | 1.4 | 0.79 |
Millan et al. (1995)
|
|
Pimozide | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 2.4 | 3.7 | 0.65 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 9.8 | 11 | 0.89 |
Sokoloff et al. (1992)
|
| [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 0.72 | 0.53 | 1.4 |
Malmberg et al. (1993)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 0.39 | 0.39 | 1.0 |
Freedman et al. (1994)
|
|
(+)-AJ76 | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 270 | 91 | 3.0 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 311 | 139 | 2.2 |
Sokoloff et al. (1992)
|
| [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 80 | 35 | 2.3 |
Malmberg et al. (1993)
|
| [125I]iodosulpiride | rStriatum | rCerebellar lob.X | 3881-b
| 1431-b
| 2.4 |
Levant et al. (1995)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 154 | 70 | 2.2 |
Millan et al. (1995)
|
|
(+)-UH232 | [125I]iodosulpiride | rD2/CHO | rD3/CHO | 40 | 9.2 | 4.3 |
Sokoloff et al. (1990)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 36 | 11 | 3.3 |
Sokoloff et al. (1990)
|
| [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 14 | 2.9 | 4.8 |
Malmberg et al. (1993)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 9.0 | 4.9 | 1.8 |
Freedman et al. (1994)
|
| [125I]iodosulpiride1-a
| rStriatum | rCerebellar lob.X | 561-b
| 231-b
| 2.4 |
Levant et al. (1995)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 125 | 215 | 0.58 |
Flietstra and Levant (1996)
|
|
(+)-Butaclamol | [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 22 | 245 | 0.090 |
Levant and De Souza (1993)
|
| [125I]iodosulpiride | hD2S/CHO | hD3/CHO | 0.44 | 2.1 | 0.21 |
Freedman et al. (1993)
|
| [3H]spiperone | hD2/CHO-K1 | hD3/CHO-K1 | 3.0 | 4.0 | 0.75 |
MacKenzie et al. (1994)
|
| [3H]spiperone | hD2/CCL1.3 | hD3/CCL1.3 | 0.69 | 11 | 0.063 |
MacKenzie et al. (1994) Tang et al. (1994)
|
| [3H]spiperone | rD2L/MN9D | hD3/MN9D | 2.6 | 4.1 | 0.63 |
Tang et al. (1994)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 0.63 | 0.22 | 2.9 |
Kula et al. (1994)
|
| [125I]NCQ-298 | hD2L/HEK 293 | rD3/HEK 293 | 0.20 | 3.2 | 0.063 |
Burris et al. (1995) |
| [125I]7-OH-PIPAT | hD2L/HEK 293 | rD3/HEK 293 | 0.69 | 5.0 | 0.14 |
Burris et al. (1995)
|
| [3H]N-0437 | hD2L/CHO-K1 | hD3/CHO-K1 | 0.42 | 1.0 | 0.42 |
Pugsley et al. (1995)
|
|
Eticlopride | [3H]spiperone | hD2/CCL1.3 | hD3/CCL1.3 | 0.07 | 0.16 | 0.44 |
MacKenzie et al. (1994) Tang et al. (1994)
|
| [3H]spiperone | rD2L/MN9D | hD3/MN9D | 0.029 | 0.46 | 0.063 |
Tang et al. (1994)
|
| [3H]YM-09151-2 | rStriatum | hD3/CCL1.3 | 0.062 | 0.043 | 1.4 |
Kula et al. (1994)
|
|
YM-09151-2 | [3H]spiperone | hD2/CCL1.3 | hD3/CCL1.3 | 0.02 | 0.06 | 0.33 |
MacKenzie et al. (1994) Tang et al. (1994)
|
| [3H]spiperone | rD2L/MN9D | hD3/MN9D | 0.03 | 0.05 | 0.60 |
Tang et al. (1994)
|
|
Risperidone | [3H]raclopride | hD2L/Ltk- | hD3/Ltk- | 1.7 | 6.7 | 0.25 |
Malmberg et al. (1993)
|
| [125I]iodosulpiride | hD2/CHO | hD3/CHO | 3.6 | 11 | 0.33 |
Millan et al. (1995)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 3.3 | 103 | 0.032 |
Flietstra and Levant (1996)
|
|
1-Nafadotride | [125I]iodosulpiride | hD2L/CHO | hD3/CHO | 3.0 | 0.31 | 9.7 |
Sautel et al. (1995b)
|
| [3H]quinpirole1-a
| rStriatum | rCerebellar lob.X | 7.0 | 3.0 | 2.3 |
Fliestra and Levant (1996)
|
|
(+)-S 14297 | [125I]iodosulpiride | hD2/CHO | hD3/CHO | 297 | 13 | 23 |
Millan et al. (1995)
|