Parameter | Entacapone (200 mg) | Tolcapone (200 mg) | Reference |
---|---|---|---|
AUC | +23% | +32% | Ruottinen and Rinne, 1996a |
Tohgi et al., 1995 | |||
+29% | +51% | Ruottinen and Rinne, 1996b | |
Davis et al., 1995a | |||
+38% | +53%6-a | Kaakkola et al., 1994b | |
Roberts et al., 1993b | |||
+46% | +58% | Myllylä et al., 1993 | |
Limousin et al., 1995 | |||
+48% | Nutt et al., 1994 | ||
T 1/2el | +17%6-a | +32%6-a | Ruottinen and Rinne, 1996b |
Roberts et al., 1993b | |||
+32% | +77% | Myllylä et al., 1993 | |
Tohgi et al., 1995 | |||
+39% | +79% | Ruottinen and Rinne, 1996a | |
Limousin et al., 1995 | |||
+75% | Nutt et al., 1994 |
↵6-a 400 mg.