Species | Tissue | Parameter Determined | Drug without Effect | Effect of Receptor Activation | Receptor Subtype | Reference |
---|---|---|---|---|---|---|
Rat | Mesenteric artery | NA release | Inhibition | A1 | Shinozuka et al., 2001 | |
Guinea pig | Vas deferens | ejp | Inhibition | A1 | Hardy and Brock, 1999 | |
Rat | Pancreas | NA release | CGS 21680 | Inhibition | A1 | Koch et al., 1998 |
Rat | Heart | NA release | CPCA | Inhibition | A1 | Snyder et al., 1998 |
Rabbit | Iris/ciliary body | NA release | CV1808 | Inhibition | A1 | Crosson and Gray, 1997 |
Rat | SCG neurons | NA release | Inhibition | P1 | Koh and Hille, 1997 | |
Human | Atrium | NA release | Inhibition | P1 | Munch et al., 1996 | |
Rabbit | Ear artery | NA release | Facilitation | P1 | Ishii et al., 1996 | |
Rat | Tail artery | NA release | Inhibition | A1 | Goncalves and Queiroz, 1996 | |
Facilitation | A2A | |||||
Rat | Caudal artery | NA release | Inhibition | P1 | Shinozuka et al., 1995 | |
Dog | Pulmonary artery | NA release | Inhibition | A1 | Vaz-da-Silva et al., 1995 | |
Guinea pig | Atrium | NA release | CGS 21680 | Inhibition | A1 | Nakatsuka et al., 1995 |
Rat | Thymus | NA release | Inhibition | P1 | Hasko et al., 1995 | |
Guinea pig | Vas deferens | NA and ATP release and neurogenic contraction | Inhibition | A1 | Driessen et al., 1994 | |
Rabbit | Ear artery | NA release | Facilitation | A1 | Maynard and Burnstock, 1994 | |
Mouse | Vas deferens | NA release | Inhibition | A1 | Kurz et al., 1993 | |
Rat | Vas deferens | NA release | Inhibition | A1 |
NA, noradrenaline; ejp, excitatory junction potential; CGS 21680, 2-p-(2-carboxyethyl)-phenethylamino-5′-N-ethylcarboxamido-adenosine; CPCA, cyclopropylcarboxamidoadenosine; CV1808, 2-phenylaminoadenosine.