CB1 and CB2 Ki values of stereoisomers of cannabidiol and of two cannabidiol analogs
| Ligand | CB1Ki Value | CB2Ki Value | Reference |
|---|---|---|---|
| nM | |||
| (−)-CBD | 4,350 | 2,860 | Showalter et al., 1996 |
| >10,000 | >10,000 | Bisogno et al., 2001 | |
| (+)-CBD | 842 | 203 | Bisogno et al., 2001 |
| (−)-5′-DMH-CBD | >10,000 | 1,800 | Bisogno et al., 2001 |
| (+)-5′-DMH-CBD | 17.4 | 211 | Bisogno et al., 2001 |
| (−)-7-OH-5′-DMH-CBD | 4,400 | 671 | Bisogno et al., 2001 |
| (+)-7-OH-5′-DMH-CBD | 2.5 | 44 | Bisogno et al., 2001 |
DMH, dimethylheptyl.