Prodrug | Drug | Pharmacology | Reference |
---|---|---|---|
5-Ethynyl-2(1H)-pyrimidinone | 5-Ethynyluracil | Mechanism-based inhibitor of DPD | Porter et al., 1994 |
IPdR | IUdR | Radiosensitizer | Kinsella et al., 1994 |
5-FP | 5-FU | Thymidylate synthase inhibitor/incorporated into DNA and RNA | Guo et al., 1995 |