Neurotoxin receptor site 1 | Tetrodotoxin | IS2–S6, IIS2–S6 |
| Saxitoxin | IIIS2–S6, IVS2–S6 |
| μ-Conotoxin | |
Neurotoxin receptor site 2 | Veratridine | IS6, IVS6 |
| Batrachotoxin | |
| Grayanotoxin | |
Neurotoxin receptor site 3 | α-Scorpion toxins | IS5–IS6, IVS3–S4 |
| Sea anemone toxins | IVS5–S6 |
Neurotoxin receptor site 4 | β-Scorpion toxins | IIS1–S2, IIS3–S4 |
Neurotoxin receptor site 5 | Brevetoxins | IS6, IVS5 |
| Ciguatoxins | |
Neurotoxin receptor site 6 | δ-Conotoxins | IVS3–S4 |
Local anesthetic receptor site | Local anesthetic drugs | IS6, IIIS6, IVS6 |
| Antiarrhythmic drugs | |
| Antiepileptic drugs |
|