Examples of receptors that demonstrate biased agonism
| Receptor | Reference |
|---|---|
| PACAP-1 | Spengler et al., 1993; Van Rampelbergh et al., 1996 |
| Dopamine D2 | Meller et al., 1992; Cordeaux et al., 2001; Mottola et al., 2002; Gay et al., 2004; Urban et al., 2007 |
| Dopamine D1 | Ryman-Rasmussen et al., 2005 |
| Histamine H3 | Krueger et al., 2005 |
| Muscarinic acetylcholine receptor | Akam et al., 2001; Thomas et al., 2008 |
| GLP-1 | Jorgensen et al., 2007 |
| Neurokinin1 | Sagan et al., 1999 |
| β2-Adrenoceptor | Seifert et al., 1999; Wenzel-Seifert and Seifert, 2000; Azzi et al., 2003; Galandrin et al., 2008 |
| PTH | Takasu et al., 1999; Bisello et al., 2002; Gesty-Palmer et al., 2006 |
| Gonadotropin-releasing receptor | Lu et al., 2007 |
| Calcitonin | Watson et al., 2000 |
| Adenosine A1 | Cordeaux et al., 2000 |
| Adenosine A3 | Gao and Jacobson, 2008 |
| δ-Opioid | Keith et al., 1998; Allouche et al., 1999; Whistler et al., 1999; Arttamangkul et al., 2008 |
| 5-HT2C | Berg et al., 1998; Werry et al., 2005 |
| 5-HT2A | Kurrasch-Orbaugh et al., 2003 |
| Cannabinoid | Bonhaus et al., 1998; Mukhopadhyay and Howlett, 2005; Shoemaker et al., 2005; Bosier et al., 2008 |
| Protease-activated receptor 1 | McLaughlin et al., 2005 |
| Chemokine CXCR2 | Hall et al., 1999 |
| α2A-Adrenoceptor | Kukkonen et al., 2001; Vilardaga et al., 2005; Nikolaev et al., 2006 |
| Bombesin | MacKinnon et al., 2001 |
| Metabotropic glutamate | Tateyama and Kubo, 2006 |
| Chemokine CCR7 | Kohout et al., 2004 |
| Angiotensin IA | Wei et al., 2003; Hunton et al., 2005 |
| Somatostatin | Liu et al., 2005; Cescato et al., 2006; Engström et al., 2006 |
| Corticotropin-releasing factor type 1 receptor | Beyermann et al., 2007 |
| CCR5 | Oppermann et al., 1999; Proudfoot et al., 1999; Watson et al., 2005 |
| Melanocortin 4 receptor | Nickolls et al., 2005 |