Enhancement of activation | | | | |
Glycine (native) | Yes | Nanomolar | Yes | Nanomolar |
Glycine α1, α1β1 | Yes | Nanomolar | Yes | Nanomolar |
Glycine α1β | Yes | Nanomolar | Yes | Micromolar |
NMDA | Yesa | Nanomolar or micromolar | Yesb | Micromolar |
Inhibition of activation | | | | |
5-HT3 | Yesc | Nanomolar | Yesc | Nanomolar |
Acetylcholine (nicotinic) | Yesc | Nanomolar | Yesc | Nanomolar or micromolar |
Glycine (native) | Yes | Nanomolar or micromolar | No | Nanomolar |
Glycine α1, α1β | No | Nanomolar | Yes | Micromolar |
Glycine α2, α3 | No | Micromolar | Yes | Nanomolar or micromolar |
Radioligand binding (↓) | | | | |
Benzodiazepine | No | Micromolar | Yes | Micromolar |