TABLE 3

Dopamine receptor agonists and antagonists that have been used clinically

The table was compiled from information presented in articles cited in the text and from the references cited therein.

DrugsMajor Clinical Application
Dopamine agonists
    ApomorphinePD, erectile dysfunction
    BromocriptinePD, pituitary tumors, hyperprolactinemia, type 2 diabetes
    CabergolinePituitary tumors, hyperprolactinemia
    FenoldopamHypertension
    PramipexolePD, restless legs syndrome, bipolar disorder, depression
    PiribedilPD
    PergolidePD
    RopinirolePD, restless legs syndrome
    RotigotinePD, bipolar disorder and depression
Dopamine antagonists
    AmisulprideSchizophrenia, bipolar disorder, depression
    AripiprazoleSchizophrenia, bipolar disorder, depression
    BenperidolSchizophrenia
    BromoprideNausea, gastroparesis
    ChlorpromazineSchizophrenia
    ClopenthixolSchizophrenia
    ClozapineSchizophrenia
    DomperidoneNausea
    DroperidolSchizophrenia, nausea
    FluphenazineSchizophrenia
    FlupentixolSchizophrenia, depression
    FluspirileneSchizophrenia
    HaloperidolSchizophrenia
    QuetiapineSchizophrenia, bipolar disorder, depression
    MetoclopramideNausea, gastroparesis
    OlanzapineSchizophrenia, bipolar disorder, depression
    PenfluridolSchizophrenia
    PerazineSchizophrenia
    PerphenazineSchizophrenia
    PimozideSchizophrenia
    ProchlorperazineSchizophrenia, nausea
    PromazineSchizophrenia
    RisperidoneSchizophrenia, bipolar disorder
    RemoxiprideSchizophrenia
    SertindoleSchizophrenia
    SulpirideSchizophrenia, depression
    SultoprideSchizophrenia
    ThiethylperazineNausea
    ThiothixeneSchizophrenia
    ThioridazineSchizophrenia
    TiaprideSchizophrenia
    TrifluperidolSchizophrenia
    TriflupromazineSchizophrenia, nausea
    TrifluoperazineSchizophrenia
    ZiprasidoneSchizophrenia, bipolar disorder, depression