Acebutolol | Diacetolol | 0.88 | 0.92 |
Albendazole | Albendazole sulfoxide | 0.10 | 0.35 |
Amitriptyline | Nortriptyline | 0.05 | 0.08 |
Amitriptyline | E-10-Hydroxynortriptyline | 0.05 | 0.31 |
Artesunate | Dihydroartimisinin | 0.25 | 0.18 |
Carbamazepine | Carbamazepine-10,11-epoxide | 0.14 | 0.33 |
Carisoprodol | Meprobamate | 0.42 | 0.76 |
Chlordiazepoxide | Demoxepam | 0.07 | 0.22 |
Chloroquine | Desethylchloroquine | 0.42 | 0.60 |
Citalopram | Desmethylcitalopram | 0.20 | 0.20 |
Citalopram | Didesmethylcitalopram | 0.20 | 0.20 |
Clobazam | N-Desemethylclobazam | 0.15 | 0.30 |
Clozapine | Norclozapine | 0.06 | 0.10 |
Codeine | Morphine | 0.93 | 0.74 |
Dasatinib | N-Dealkyldasatinib | 0.04 | 0.07 |
Desipramine | 2-Hydroxydesipramine | 0.10 | 0.20 |
Desloratadine | 3-Hydroxydesloratadine | 0.15 | 0.13 |
Diazepam | Desmethyldiazepam | 0.023 | 0.03 |
Diazepam | Temazepam | 0.023 | 0.038 |
Diazepam | Oxazepam | 0.023 | 0.04 |
Diltiazem | Desacetyldiltiazem | 0.25 | 0.23 |
Diltiazem | N-Desmethyldiltiazem | 0.25 | 0.32 |
Disopyramide | N-Desisopropyldisopyramide | 0.35–0.95 | 0.90–0.95 |
Doxepin | Desmethyldoxepin | 0.20 | 0.21 |
Flutamide | 2-Hydroxyflutamide | 0.05 | 0.07 |
Hydroxyzine | Cetirizine | 0.07 | 0.07 |
Imatinib | N-Desmethylimatinib | 0.05 | 0.05 |
Imipramine | Desipramine | 0.03 | 0.11 |
Imipramine | 2-Hydroxydesipramine | 0.03 | 0.20 |
Ketamine | Norketamine | 0.40 | 0.50 |
Levosimendan | Or-1896 | 0.02 | 0.60 |
Lidocaine | Monoethyl glycine xylidide (MEGX) | 0.45 | 0.86 |
Lidocaine | Glycine xylidide (GX) | 0.45 | 0.95 |
Loratadine | Desloratadine | 0.03 | 0.15 |
Losartan | Exp3174 | 0.013 | 0.002 |
Loxapine | Amoxapine | NA | 0.10 |
Meperidine | Normeperidine | 0.56 | 0.66 |
Midazolam | 1′-Hydroxymidazolam | 0.02 | 0.11 |
Midazolam | 1′-Hydroxymidazolam glucuronide | 0.02 | 0.57 |
Morphine | Morphine-6-glucuronide | 0.74 | 0.89 |
Nortriptyline | 10-Hydroxynortriptyline | 0.08 | 0.31 |
Oxcarbazepine | 10-Hydroxycarbamazepine | 0.41 | 0.61 |
Oxybutynin | Desethyloxybutynin | 0.0034 | 0.0018 |
Pioglitazone | Ketopioglitazone | 0.016 | 0.02 |
Pioglitazone | Hydroxypioglitazone | 0.016 | 0.02 |
Primidone | Phenobarbital | 0.70 | 0.72 |
Procainamide | N-Acetylprocainamide | 0.84 | 0.90 |
Propafenone | 5-Hydroxypropafenone | 0.08 | 0.12 |
Propoxyphene | Norpropoxyphene | 0.24 | 0.26 |
Quinidine | 3-Hydroxyquinidine | 0.13 | 0.40 |
Risperidone | Paliperidone | 0.10 | 0.23 |
Roflumilast | Roflumilast N-oxide | 0.01 | 0.03 |
Sibutramine | Desmethylsibutramine | 0.03 | 0.06 |
Sibutramine | Didesmethylsibutramine | 0.03 | 0.06 |
Spironolactone | Canrenone | 0.06 | 0.02 |
Terfenadine | Fexofenadine | 0.05 | 0.35 |
Thioridazine | Sulforidazine | 0.0016 | 0.017 |
Thioridazine | Mesoridazine | 0.0016 | 0.017–0.09 |
Tolterodine | Desfesoterodine | 0.037 | 0.36 |
Triamterene | 4-Hydroxytriamterene sulfate | 0.39 | 0.10 |
Trimethadione | Dimethadione | 0.91 | 0.94 |
Valproic acid | 2-Propyl-2-Pentenoic acid | 0.10 | 0.007 |
Venlafaxine | Desvenlafaxine | 0.73 | 0.70 |
Verapamil | Norverapamil | 0.10 | 0.13 |