Receptor | Ligand | EC50 | Readout | System | Reference |
---|---|---|---|---|---|
nM | |||||
mMRGPRA1 | FMRFamide | 20 | calcium | HEK293-Gα15 | Dong et al., 2001 |
NPFF | 200 | calcium | HEK293-Gα15 | Dong et al., 2001 | |
hβ-Salusin | 300 | calcium | HEK293 | Wang et al., 2006b | |
chloroquine | 300,000 | calcium | HEK293 | Liu et al., 2009 | |
mMRGPRA4 | NPAF | 60 | calcium | HEK293-Gα15 | Dong et al., 2001 |
mMRGPRA3 | chloroquine | 27,000 | calcium | HEK293 | Liu et al., 2009 |
rMRGPRA | chloroquine | N.D. | calcium | mDRG neurons | Liu et al., 2009 |
adenine | 3 | cAMP inhibition | CHO | Bender et al., 2002 | |
60 | GTPγS | CHO | Bender et al., 2002 |
GTPγS, guanosine 5′-3-O-(thio)triphosphate; N.D., not determined; r, rat; m, mouse.