TABLE 2

Amino acid residues of galanin receptors involved in ligand binding found by docking studies

ReceptorResidues
GAL1aGln92, Val95, Tyr96, Cys108, His112, Phe115, Thr116, Met119, Cys203, Val206, His263, His264, His267, Ile286, His289
GAL2aGln82, Ile105, Phe106, Met109, Tyr160, Tyr163, Tyr164, Asn171, Thr173, Asp188, Thr191, Ser195, His253, Ile256, His278, Tyr282
GAL3a,bGln79a,b, Ile82a,b, Asp86b, Trp88b, Cys95a, Val98a, His99a,b, Ile102a,b, Tyr103a,b, Tyr161a, Tyr166a, Glu170b, Pro174b, Ala175b, Asp185b, His251a, Tyr270a, Arg273a,b, His277a,b, Tyr281a
  • a Jurkowski et al. (2013).

  • b Kothandan et al. (2013).