OCT1 | SLC | SLC22 | SLC22A1 | — | Metformin, oxaliplatin |
OCT2 | SLC | SLC22 | SLC22A2 | — | Metformin, ranitidine, varinicline |
OCT3 | SLC | SLC22 | SLC22A3 | R-S-H-L | Histamine, epinephrine |
OCTN1 | SLC | SLC22 | SLC22A4 | L-T-A-F | Quinidine, verapamil, ipratropium, ergothioneine |
OCTN2 | SLC | SLC22 | SLC22A5 | S-T-A-F | Carnitine, amisulpride, cephaloridine |
OAT1 | SLC | SLC22 | SLC22A6 | — | Lamivudine, acyclovir, ciprofloxacin |
OAT2 | SLC | SLC22 | SLC22A7 | — | Bumetanide, erythromycin, paclitaxel |
OAT3 | SLC | SLC22 | SLC22A8 | — | Furosemide, bumetanide |
OAT4 | SLC | SLC22 | SLC22A11 | S-T-S-L | Bumetanide, urate, methotrexate |
URAT1 | SLC | SLC22 | SLC22A12 | S-T-Q-F | Urate |
OATP1A2 | SLC | SLCO | SLCO1A2 | K-T-K-L | Statins, fexofenadine |
OATP1B1 | SLC | SLCO | SLCO1B1 | — | Statins, repaglinide, olmesartan |
OATP1B3 | SLC | SLCO | SLCO1B3 | — | Statins, telmisartan, fexofenadine |
OATP1C1 | SLC | SLCO | SLCO1C1 | E-T-Q-L | Triiodothyronine, thyroxine |
OATP2B1 | SLC | SLCO | SLCO2B1 | D-S-R-V | Statins, fexofenadine |
OATP3A1 | SLC | SLCO | SLCO3A1 | E-S-V-L | Benzylpenicillin, vasopressin |
OATP4A1 | SLC | SLCO | SLCO4A1 | Q-S-S-V | Estradiol-17β-glucuronide |
OATP4C1 | SLC | SLCO | SLCO4C1 | — | Digoxin, methotrexate, sitagliptin |
PEPT1 | SLC | SLC15 | SLC15A1 | Q-K-Q-M | Cephalexin, valacyclovir, enalapril |
PEPT2 | SLC | SLC15 | SLC15A2 | K-T-K-L | Cephalexin, valacyclovir, enalapril |
MDR1 (Pgp) | ABC | ABCB | ABCB1 | — | Digoxin, loperamide |
BCRP | ABC | ABCG | ABCG2 | — | Statins, methotrexate |
MRP1 | ABC | ABCC | ABCC1 | — | Citalopram, methotrexate, Leukotriene C4 |
MRP2 | ABC | ABCC | ABCC2 | S-T-K-F | Olmesartan, methotrexate, etoposide |
MRP3 | ABC | ABCC | ABCC3 | — | Estradiol-17β-glucuronide |
MRP4 | ABC | ABCC | ABCC4 | E-T-A-L | Adefovir, topotecan, methotrexate |
MRP7 | ABC | ABCC | ABCC10 | D-T-R-L | Docetaxel, paclitaxel, viscristine, vinblastine |