| | | μM |
TAAR3 | Rat, mouse | Cyclohexylamine | 7 (mouse),b 20 (mouse)c |
| | Isoamylamine | 10 (mouse)b,c |
| | Octylamine | 50 (mouse)b |
| | PEA | 40 (mouse)b |
TAAR4 | Rat, mouse | PEA | 0.7 (mouse),b 1 (mouse)c |
TAAR5 | Human, rat, mouse | Trimethylamine | 0.7 (mouse),b 0.3 (mouse),d 1 (rat),d 0.12 (human)e |
| | N,N-dimethylethylamine | 1 (mouse),b 0.17 (human)e |
| | N,N-dimethyloctylamine | 1 (mouse)b |
| | N-methylpiperidine | 3 (mouse),b 20 (mouse),c >10 (human)e |
| | Pyrrolidine | 17 (mouse)b |
| | Triethylamine | 22 (mouse)b |
| | 3-pyrroline | 42 (mouse)b |
| | 2-methy-1-pyrroline | 46 (mouse)b |
| | 3ITa | 4.4 (human)f |
TAAR7b | Rat, mouse | N,N-dimethyloctylamine | 3 (mouse)b |
| | N,N-dimethylbutylamine | 30 (mouse)b |
TAAR7e | Rat, mouse | Octylamine | 28 (mouse)b |
| | Heptylamine | 34 (mouse)b |
| | 2-methy-1-pyrroline | 48 (mouse)b |
TAAR7d | Rat, mouse | N,N-dimethylcyclohexylamine | 0.5 (mouse)b |
| | N-methylpiperidine | 16 (mouse)b |
| | N,N-dimethylbutylamine | 30 (mouse)b |
| | 1-(2-aminoethyl)piperidine | 30 (mouse)b |
| | Heptylamine | 33 (mouse)b |
| | 2-methy-1-pyrroline | 50 (mouse)b |
TAAR8c | Human, rat, mouse | N-methylpiperidine | 0.5 (rat)g |
| | N,N-dimethylcyclohexylamine | 13 (rat)g |
TAAR9 | Human, rat, mouse | N-methylpiperidine | 18 (rat)g |
| | N,N-dimethylcyclohexylamine | 27 (rat)g |
Zebrafish TAARs | | | |
TAAR10a | Zebrafish | Serotonin | 0.5h |
| | 5-methoxytryptamine | 20h |
TAAR10b | Zebrafish | TRP | 50h |
TAAR12h | Zebrafish | β-phenyethylamine | 0.3h |
TAAR13a | Zebrafish | Histamine | 20h |
TAAR13c | Zebrafish | Cadaverine | 20,i 10h |
TAAR13d | Zebrafish | Putrescine | 1h |
TAAR16c | Zebrafish | N-methylpiperidine | 10h |
TAAR16e | Zebrafish | N,N-dimethylcyclohexylamine | 30h |