TABLE 6

Ligand-binding affinities of SST3-selective ligands

SST1SST2SST3SST4SST5
L-796/778a1255>10,0002486501200
sst3-ODN-8b>10,000>10,0004.1>10,000>10,000
ACQ090c5.685.318.136.815.93
MK-4256d236240250.66384533
  • a Data from Rohrer et al. (1998).

  • b Data from Reubi et al. (2000a).

  • c Data from Troxler et al. (2010).

  • d Data from He et al. (2012).