TABLE 8

Ligand-binding affinities of SST5-selective ligands

SST1SST2SST3SST4SST5
L-817/818a3.35264820.4
BIM-23268b18.415.161.616.30.37
S5A1c>5190>10,000>10,0004.87
  • a Data from Rohrer et al. (1998).

  • b Data from Shimon et al. (1997a).

  • c Data from Farb et al. (2017).