Rapid communicationThe first radiolabeled histamine H3 receptor antagonist, [125I]iodophenpropit: Saturable and reversible binding to rat cortex membranes
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Use of an inverse agonist radioligand [<sup>3</sup>H]A-317920 reveals distinct pharmacological profiles of the rat histamine H<inf>3</inf> receptor
2006, NeuropharmacologyCitation Excerpt :Moreover, clobenpropit and thioperamide have been reported to have significant affinities for the human histamine H4 receptor (O'Reilly et al., 2002; Esbenshade et al., 2003) that would be expected to limit their utility. Two additional radioligands, [125I]iodophenpropit (Jansen et al., 1992) and [3H]S-methylthioperamide (Yanai et al., 1994) have also been described as antagonist radioligands for the H3 histamine receptor. However, these H3 receptor radioligands exhibited lower signal to noise ratios and are also not commercially available.
The profiles of human and primate [<sup>3</sup>H]N(α)-methylhistamine binding differ from that of rodents
1999, European Journal of PharmacologyBiochemical properties of the histamine H<inf>3</inf> receptor
1998, Pharmacochemistry LibrarySynthesis of radioligands for the histamine H<inf>3</inf> receptor
1998, Pharmacochemistry LibraryMedicinal chemistry of histamine H3 receptor antagonists
1998, Pharmacochemistry Library
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