Structure-activity relationships of steroid hormones on muscarinic receptor binding
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Neurosteroids and steroid hormones are allosteric modulators of muscarinic receptors
2021, NeuropharmacologyCitation Excerpt :Steroids have been shown to improve memory by affecting acetylcholine release and cholinergic neurotransmission (Daniel et al., 2005; Darnaudéry et al., 2000; Pallarés et al., 1998). Moreover, steroid hormones may inhibit the binding of muscarinic ligands (Horishita et al., 2005; B. B. Klangkalya and Chan, 1988; Borpit Borpit Klangkalya and Chan, 1988; Wilkinson et al., 1995, 1992). However, all reports so far describe the effects of steroids on muscarinic receptors only at micromolar or higher concentrations.
Neuroactive steroids, WIN-compounds and cholesterol share a common binding site on muscarinic acetylcholine receptors
2021, Biochemical PharmacologyCitation Excerpt :NAS are known as compounds that can trigger fast, non-genomic effects via stimulation of various ligand-gated ion channels, voltage-gated ion channels, or G-protein coupled receptors [20]. Several studies have shown that NS modulate muscarinic receptors at micromolar concentrations [21–25]. In our recent study, we have shown that NS and steroid hormones at nanomolar concentrations allosterically modulate functional responses of muscarinic receptors to acetylcholine [26].
Place of pregnenolone neurosteroid in the nervous system: Physiological role and pathogenic implications
2009, Medecine et LongeviteSteroids and depression
1991, Journal of Steroid Biochemistry and Molecular BiologyContinuous stereospecific Δ<sup>4</sup>-3-keto-steroid reduction by PAAH bead-entrapped Clostridium paraputrificum cells
1990, Enzyme and Microbial Technology
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Present address: Department of Pharmacology, Pramongkutklao College of Medicine, Rajavithi Road, Bangkok, Thailand, 10400.