Molecular pharmacological aspects of histamine receptors
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2018, Neuroscience LettersCitation Excerpt :The H3 receptor is expressed mainly in structures of the central and peripheral nervous systems and has multiples isoforms [19,20], which gives it high heterogeneity [14]. The H3 receptor exerts inhibitory presynaptic activity on the synthesis and release of histamine [21,19], and alterations on its function is related to changes in behavior, metabolic syndromes [14] and locomotion [22]. The H4 receptor is found in greater amounts in peripheral tissues [14], participating in inflammatory processes, allergies and autoimmune diseases [23].
Markers of anaphylaxis – a systematic review
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2018, iScienceCitation Excerpt :Lisuride is primarily metabolized in the liver, where there is a relatively high expression of histamine receptors. There is also high receptor expression in the gastrointestinal tract owing to the role of histamine in intestinal secretion and motility (Leurs et al., 1995; Sander et al., 2006). Furthermore, lisuride administration in patients with Parkinson disease has been associated with gastrointestinal side effects (Ebadi and Pfeiffer, 2004).
Antihistamines as promising drugs in cancer therapy
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