[3H]8-Ethyl-4-methyl-2-phenyl-(8R)-4,5,7,8-tetrahydro-1H-imidazo[2,1-i]-purin-5-one ([3H]PSB-11), a Novel High-Affinity Antagonist Radioligand for Human A3 Adenosine Receptors
The preparation and preliminary evaluation of [3H]PSB-11 is described
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Acknowledgements
V.O. was supported by a Humboldt scholarship. C.E.M. is grateful for support by the Fonds der Chemischen Industrie and the Deutsche Forschungsgemeinschaft (GRK677).
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V.O. was on leave from the Latvian Institute of Organic Synthesis, Riga, Latvia, supported by a Humboldt fellowship.
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