Property-based design: optimization of drug absorption and pharmacokinetics

J Med Chem. 2001 Apr 26;44(9):1313-33. doi: 10.1021/jm000407e.
No abstract available

Publication types

  • Review

MeSH terms

  • Animals
  • Biological Transport
  • Blood Proteins / metabolism
  • Blood-Brain Barrier
  • Caco-2 Cells
  • Cell Membrane / metabolism
  • Drug Design*
  • Eye / metabolism
  • Humans
  • Intestinal Absorption
  • Models, Biological
  • Models, Molecular
  • Nasal Mucosa / metabolism
  • Pharmaceutical Preparations / metabolism*
  • Pharmacokinetics*
  • Prodrugs / metabolism
  • Skin Absorption

Substances

  • Blood Proteins
  • Pharmaceutical Preparations
  • Prodrugs