The PXR ligand-binding domain: how to be picky and promiscuous at the same time

Trends Pharmacol Sci. 2001 Sep;22(9):448. doi: 10.1016/s0165-6147(00)01847-2.
No abstract available

Publication types

  • News

MeSH terms

  • Binding Sites
  • Diphosphonates / metabolism*
  • Drug Interactions
  • Pregnane X Receptor
  • Receptors, Cytoplasmic and Nuclear / metabolism
  • Receptors, Cytoplasmic and Nuclear / physiology*
  • Receptors, Steroid / metabolism
  • Receptors, Steroid / physiology*

Substances

  • Diphosphonates
  • Pregnane X Receptor
  • Receptors, Cytoplasmic and Nuclear
  • Receptors, Steroid
  • SR 12813