Enhanced analgesic activity of D-Ala2 enkephalinamides following D-isomer substitutions at position five

Life Sci. 1978 Jul 10;23(2):99-104. doi: 10.1016/0024-3205(78)90256-4.
No abstract available

MeSH terms

  • Analgesics*
  • Animals
  • Electroshock
  • Endorphins / pharmacology*
  • Enkephalins / analysis
  • Enkephalins / pharmacology*
  • Haplorhini
  • Male
  • Morphine / pharmacology
  • Rats
  • Reaction Time / drug effects
  • Receptors, Opioid / metabolism

Substances

  • Analgesics
  • Endorphins
  • Enkephalins
  • Receptors, Opioid
  • Morphine