Conversion of a gonadotropin-releasing hormone antagonist to an agonist

Nature. 1982 Apr 15;296(5858):653-5. doi: 10.1038/296653a0.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Cells, Cultured
  • Gonadotropin-Releasing Hormone / antagonists & inhibitors*
  • Luteinizing Hormone / metabolism
  • Macromolecular Substances
  • Membrane Fluidity
  • Mice
  • Pituitary Gland / cytology
  • Receptors, Cell Surface / drug effects
  • Receptors, Cell Surface / physiology*
  • Receptors, LHRH
  • Structure-Activity Relationship

Substances

  • Macromolecular Substances
  • Receptors, Cell Surface
  • Receptors, LHRH
  • Gonadotropin-Releasing Hormone
  • Luteinizing Hormone