A chimeric vesicular monoamine transporter dissociates sensitivity to tetrabenazine and unsubstituted aromatic amines

Adv Pharmacol. 1998:42:227-32. doi: 10.1016/s1054-3589(08)60734-6.
No abstract available

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Cell Line
  • Cell Membrane / metabolism
  • Cell Membrane / ultrastructure
  • Chlorocebus aethiops
  • Histamine / pharmacology
  • Humans
  • Kinetics
  • Membrane Glycoproteins / chemistry*
  • Membrane Glycoproteins / drug effects
  • Membrane Glycoproteins / metabolism*
  • Membrane Transport Proteins*
  • Models, Structural
  • Neuropeptides*
  • Protein Conformation
  • Recombinant Fusion Proteins / chemistry
  • Recombinant Fusion Proteins / drug effects
  • Recombinant Fusion Proteins / metabolism
  • Serotonin / metabolism*
  • Tetrabenazine / pharmacology*
  • Transfection
  • Vesicular Biogenic Amine Transport Proteins
  • Vesicular Monoamine Transport Proteins

Substances

  • Membrane Glycoproteins
  • Membrane Transport Proteins
  • Neuropeptides
  • Recombinant Fusion Proteins
  • Vesicular Biogenic Amine Transport Proteins
  • Vesicular Monoamine Transport Proteins
  • Serotonin
  • Histamine
  • Tetrabenazine