Research ArticleIUPHAR Nomenclature Reports
International Union of Basic and Clinical Pharmacology. LXXIV. Apelin Receptor Nomenclature, Distribution, Pharmacology, and Function
Sarah L. Pitkin, Janet. J. Maguire, Tom I. Bonner and Anthony P. Davenport
Pharmacological Reviews September 2010, 62 (3) 331-342; DOI: https://doi.org/10.1124/pr.110.002949
Sarah L. Pitkin
Clinical Pharmacology Unit, University of Cambridge, Cambridge, United Kingdom (S.L.P., J.J.M., A.P.D.); and Section on Functional Neuroscience, National Institute of Mental Health, Bethesda, Maryland (T.I.B.)
Janet. J. Maguire
Clinical Pharmacology Unit, University of Cambridge, Cambridge, United Kingdom (S.L.P., J.J.M., A.P.D.); and Section on Functional Neuroscience, National Institute of Mental Health, Bethesda, Maryland (T.I.B.)
Tom I. Bonner
Clinical Pharmacology Unit, University of Cambridge, Cambridge, United Kingdom (S.L.P., J.J.M., A.P.D.); and Section on Functional Neuroscience, National Institute of Mental Health, Bethesda, Maryland (T.I.B.)
Anthony P. Davenport
Clinical Pharmacology Unit, University of Cambridge, Cambridge, United Kingdom (S.L.P., J.J.M., A.P.D.); and Section on Functional Neuroscience, National Institute of Mental Health, Bethesda, Maryland (T.I.B.)

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Research ArticleIUPHAR Nomenclature Reports
International Union of Basic and Clinical Pharmacology. LXXIV. Apelin Receptor Nomenclature, Distribution, Pharmacology, and Function
Sarah L. Pitkin, Janet. J. Maguire, Tom I. Bonner and Anthony P. Davenport
Pharmacological Reviews September 1, 2010, 62 (3) 331-342; DOI: https://doi.org/10.1124/pr.110.002949
Research ArticleIUPHAR Nomenclature Reports
International Union of Basic and Clinical Pharmacology. LXXIV. Apelin Receptor Nomenclature, Distribution, Pharmacology, and Function
Sarah L. Pitkin, Janet. J. Maguire, Tom I. Bonner and Anthony P. Davenport
Pharmacological Reviews September 1, 2010, 62 (3) 331-342; DOI: https://doi.org/10.1124/pr.110.002949
Jump to section
- Article
- Abstract
- I. Introduction
- II. The Apelin Receptor: Recommendations for Nomenclature
- III. Receptor Structure
- IV. Endogenous Agonists
- V. Receptor Distribution
- VI. Apelin Peptide Distribution
- VII. Synthetic Agonists
- VIII. Antagonists
- IX. Radiolabeled Ligands
- X. Physiological Roles
- XI. Pathophysiological Roles
- XII. Single-Nucleotide Polymorphisms
- XIII. Knockout Mouse Models
- XIV. Conclusion
- Acknowledgments.
- Footnotes
- References
- Figures & Data
- Info & Metrics
- eLetters
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