Research ArticleIUPHAR Nomenclature Reports
International Union of Basic and Clinical Pharmacology. LXXV. Nomenclature, Classification, and Pharmacology of G Protein-Coupled Melatonin Receptors
Margarita L. Dubocovich, Philippe Delagrange, Diana N. Krause, David Sugden, Daniel P. Cardinali and James Olcese
Pharmacological Reviews September 2010, 62 (3) 343-380; DOI: https://doi.org/10.1124/pr.110.002832
Margarita L. Dubocovich
Department of Pharmacology and Toxicology, School of Medicine and Biomedical Sciences, University at Buffalo, State University of New York, Buffalo, New York (M.L.D.); Department Molecular Pharmacology and Biological Chemistry, Feinberg School of Medicine, Northwestern University, Chicago, Illinois (M.L.D.); Experimental Sciences Department, Institut de Recherches Servier, Suresnes, France (P.D.); Department of Pharmacology, College of Medicine, University of California, Irvine, California (D.N.K.); Division of Reproduction and Endocrinology, School of Biomedical and Health Sciences, King's College London, United Kingdom (D.S.); Department of Teaching & Research, Faculty of Medical Sciences, Pontificia Universidad Católica Argentina, Buenos Aires, Argentina (D.P.C.); and Department of Biomedical Sciences, Florida State University College of Medicine, Tallahassee, Florida (J.O.)
Philippe Delagrange
Department of Pharmacology and Toxicology, School of Medicine and Biomedical Sciences, University at Buffalo, State University of New York, Buffalo, New York (M.L.D.); Department Molecular Pharmacology and Biological Chemistry, Feinberg School of Medicine, Northwestern University, Chicago, Illinois (M.L.D.); Experimental Sciences Department, Institut de Recherches Servier, Suresnes, France (P.D.); Department of Pharmacology, College of Medicine, University of California, Irvine, California (D.N.K.); Division of Reproduction and Endocrinology, School of Biomedical and Health Sciences, King's College London, United Kingdom (D.S.); Department of Teaching & Research, Faculty of Medical Sciences, Pontificia Universidad Católica Argentina, Buenos Aires, Argentina (D.P.C.); and Department of Biomedical Sciences, Florida State University College of Medicine, Tallahassee, Florida (J.O.)
Diana N. Krause
Department of Pharmacology and Toxicology, School of Medicine and Biomedical Sciences, University at Buffalo, State University of New York, Buffalo, New York (M.L.D.); Department Molecular Pharmacology and Biological Chemistry, Feinberg School of Medicine, Northwestern University, Chicago, Illinois (M.L.D.); Experimental Sciences Department, Institut de Recherches Servier, Suresnes, France (P.D.); Department of Pharmacology, College of Medicine, University of California, Irvine, California (D.N.K.); Division of Reproduction and Endocrinology, School of Biomedical and Health Sciences, King's College London, United Kingdom (D.S.); Department of Teaching & Research, Faculty of Medical Sciences, Pontificia Universidad Católica Argentina, Buenos Aires, Argentina (D.P.C.); and Department of Biomedical Sciences, Florida State University College of Medicine, Tallahassee, Florida (J.O.)
David Sugden
Department of Pharmacology and Toxicology, School of Medicine and Biomedical Sciences, University at Buffalo, State University of New York, Buffalo, New York (M.L.D.); Department Molecular Pharmacology and Biological Chemistry, Feinberg School of Medicine, Northwestern University, Chicago, Illinois (M.L.D.); Experimental Sciences Department, Institut de Recherches Servier, Suresnes, France (P.D.); Department of Pharmacology, College of Medicine, University of California, Irvine, California (D.N.K.); Division of Reproduction and Endocrinology, School of Biomedical and Health Sciences, King's College London, United Kingdom (D.S.); Department of Teaching & Research, Faculty of Medical Sciences, Pontificia Universidad Católica Argentina, Buenos Aires, Argentina (D.P.C.); and Department of Biomedical Sciences, Florida State University College of Medicine, Tallahassee, Florida (J.O.)
Daniel P. Cardinali
Department of Pharmacology and Toxicology, School of Medicine and Biomedical Sciences, University at Buffalo, State University of New York, Buffalo, New York (M.L.D.); Department Molecular Pharmacology and Biological Chemistry, Feinberg School of Medicine, Northwestern University, Chicago, Illinois (M.L.D.); Experimental Sciences Department, Institut de Recherches Servier, Suresnes, France (P.D.); Department of Pharmacology, College of Medicine, University of California, Irvine, California (D.N.K.); Division of Reproduction and Endocrinology, School of Biomedical and Health Sciences, King's College London, United Kingdom (D.S.); Department of Teaching & Research, Faculty of Medical Sciences, Pontificia Universidad Católica Argentina, Buenos Aires, Argentina (D.P.C.); and Department of Biomedical Sciences, Florida State University College of Medicine, Tallahassee, Florida (J.O.)
James Olcese
Department of Pharmacology and Toxicology, School of Medicine and Biomedical Sciences, University at Buffalo, State University of New York, Buffalo, New York (M.L.D.); Department Molecular Pharmacology and Biological Chemistry, Feinberg School of Medicine, Northwestern University, Chicago, Illinois (M.L.D.); Experimental Sciences Department, Institut de Recherches Servier, Suresnes, France (P.D.); Department of Pharmacology, College of Medicine, University of California, Irvine, California (D.N.K.); Division of Reproduction and Endocrinology, School of Biomedical and Health Sciences, King's College London, United Kingdom (D.S.); Department of Teaching & Research, Faculty of Medical Sciences, Pontificia Universidad Católica Argentina, Buenos Aires, Argentina (D.P.C.); and Department of Biomedical Sciences, Florida State University College of Medicine, Tallahassee, Florida (J.O.)
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Research ArticleIUPHAR Nomenclature Reports
International Union of Basic and Clinical Pharmacology. LXXV. Nomenclature, Classification, and Pharmacology of G Protein-Coupled Melatonin Receptors
Margarita L. Dubocovich, Philippe Delagrange, Diana N. Krause, David Sugden, Daniel P. Cardinali and James Olcese
Pharmacological Reviews September 1, 2010, 62 (3) 343-380; DOI: https://doi.org/10.1124/pr.110.002832
Research ArticleIUPHAR Nomenclature Reports
International Union of Basic and Clinical Pharmacology. LXXV. Nomenclature, Classification, and Pharmacology of G Protein-Coupled Melatonin Receptors
Margarita L. Dubocovich, Philippe Delagrange, Diana N. Krause, David Sugden, Daniel P. Cardinali and James Olcese
Pharmacological Reviews September 1, 2010, 62 (3) 343-380; DOI: https://doi.org/10.1124/pr.110.002832
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- Article
- Abstract
- I. Introduction
- II. G Protein-Coupled Melatonin Receptor Family
- III. Cellular Signaling of MT1 and MT2 Melatonin Receptors
- IV. MT1 and MT2 Melatonin Receptors: Structure-Activity Relationships and Selective Ligands
- V. MT1- and MT2-Mediated Functional Responses
- VI. Melatonin receptors as therapeutic targets
- VII. Conclusion
- Acknowledgments.
- Footnotes
- References
- Figures & Data
- Info & Metrics
- eLetters
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