Inhibitor | Ki | Application | Binding Site Model | |
---|---|---|---|---|
GLYT1 | GLYT2 | |||
nM | ||||
GLYT1 inhibitors | ||||
Sarcosinea,b | 55,000 | >100,000 | Pharmacological tool | |
NFPS (ALX 5407)c | 3 | >1000 | Pharmacological tool | |
ORG 24598b | 32 | >100,000 | Pharmacological tool | |
LY2365109d | 15.8 | >30,000 | Pharmacological tool | |
GLY2 inhibitors | ||||
ORG 25543e | >100 | 16 | Pharmacological tool | |
N-Arachidonylglycinef | >100,000 | 3000 | Pharmacological tool | Edington et al., 2009 |