Receptor | Ligand | KD | Tissue |
---|---|---|---|
H1-receptor | [3H]Mepyramine | 0.8 nm | Guinea pig brain7-a |
[125I]Iodobolpyramine | 0.1 nm | Guinea pig brain7-b | |
[125I]Iodoazidophenpyramine | 0.01 nm | Guinea pig cerebellum7-c | |
[11C]Mepyramine | 1.0 nm | Human brain (in vivo)7-d | |
[11C]Doxepin | 0.1 nm | Human brain (in vivo)7-e | |
H2-receptor | [3H]Tiotidine | 25 nm | Guinea pig brain7-f |
[125I]Iodoaminopotentidine | 0.3 nm | Guinea pig brain7-g | |
[125I]Iodoazidopotentidine | 10 nm | Guinea pig brain7-g | |
H 3-receptor | [3H]R-(α)-methylhistamine | 0.5 nm | Rat brain7-h |
[3H]Nα-methylhistamine | 2.0 nm | Rat cerebral cortex7-i | |
[125I]Iodophenpropit | 0.3 nm | Rat cerebral cortex7-j | |
[125I]Iodoproxyfan | 0.065 nm | Rat striatum7-k | |
[3H]GR168320 | 0.1 nm | Rat cerebral cortex7-l |
↵7-a Hill et al. (1981)
↵7-b Körner et al. (1986)
↵7-c Ruat et al. (1988)
↵7-d Villemagne et al. (1991)
↵7-e Yanai et al. (1995)
↵7-f Gajtkowski et al. (1983)
↵7-g Ruat et al. (1990a)
↵7-h Arrang et al. (1990)
↵7-i Clark and Hill (1995)
↵7-j Jansen et al. (1992)
↵7-k Ligneau et al. (1994)
↵7-l Brown et al. (1994)