Species | Tissue | Effect of Receptor Activation | Receptor Subtype | Agonists | Antagonists | Drugs without Effect | Reference |
---|---|---|---|---|---|---|---|
Rat | Mesenteric artery | Inhibition | P2 | β,γ-MeATP2-a | DPCPX2-b | Shinozuka et al., 2001 | |
2MeSATP2-c | PPADS2-d | ||||||
Guinea pig | Atrium | Stimulation | P2X3 | ATP | PPADS | Reactive blue 2 | Sperlagh et al., 2000 |
Facilitation | 2MeSATP | Suramin | |||||
α,β-MeATP2-e | TNP-ATP2-f | ||||||
β,γ-MeATP | |||||||
ADP | |||||||
Rat | Cultured sympathetic neurons | Stimulation | P2X | ATP | Suramin | DIDS | von Kugelgen et al., 1999b |
Cibacron blue 3GA | |||||||
Rat | Cultured sympathetic neurons | Stimulation | P2X2 | ATP | Suramin | ADP | Boehm, 1999 |
Facilitation | 2MeSATP | PPADS | UDP | ||||
ATPγS2-g | α,β-MeATP | ||||||
β,γ-MeATP | |||||||
Rabbit | Ear artery | Facilitation | P2Y | β,γ-MeATP | Ishii-Nozawa et al., 1999 | ||
Rat | Pancreas | Inhibition | P2Y | ATP | Cibacron blue 3GA | PPADS | Koch et al., 1998 |
ATPγS | Reactive blue 2 | ||||||
ADPβS | Reactive red 2 | ||||||
Rat | Kidney | Inhibition | P2Y | ATPγS | Cibacron blue 3GA | Suramin | Bohmann et al., 1997 |
Rat | Tail artery | Inhibition | P2Y | 2MeSATP | Cibacron blue 3GA | Goncalves and Queiroz, 1996 | |
Suramin | |||||||
Rabbit | Ear artery | Facilitation | Neither P1 nor P2 | β,γ-MeATP | α,β-MeATP | Ishii et al., 1995 | |
ATP | |||||||
2MeSATP | |||||||
Rat | Atrium | Inhibition | P2Y | ATPγS | Cibacron blue 3GA | β,γ-Me-l-ATP | von Kugelgen et al., 1995 |
ATP | |||||||
Chicken | Sympathetic neurons | Facilitation | P2 | ATP | Reactive blue 2 | Allgaier et al., 1995a | |
2MeSATP | Suramin | ||||||
Inhibition | P2 | ATP | Suramin | Reactive blue 2 | |||
Chicken | Sympathetic neurons | Inhibition | P2 | ATP | Suramin | Allgaier et al., 1994a | |
Facilitation | P2Y | 2MeSATP | Suramin | α,β-MeATP | |||
Rabbit | Vas deferens | Inhibition | P3 | ATP | α,β-MeATP | Todorov et al., 1994 | |
β,γ-MeATP | |||||||
Adenosine | |||||||
2-Chloroadenosine | |||||||
Saphenous artery | Facilitation | P3 | ATP | 8-SPT2-h | α,β-MeATP | ||
β,γ-MeATP | |||||||
Adenosine | |||||||
2-Chloroadenosine | |||||||
Mouse | Vas deferens | Inhibition | P2Y | ATPγS | Reactive blue 2 | von Kugelgen et al., 1994b | |
Brilliant blue G | |||||||
Suramin | |||||||
PPADS | |||||||
Rat | Vas deferens | Inhibition | P2Y | Reactive blue 2 | |||
Brilliant blue G | |||||||
Suramin | |||||||
Mouse | Vas deferens | Inhibition | P2Y | α,β-MeATP | Suramin | Kurz et al., 1993 | |
β,γ-MeATP | |||||||
2MeSATP | |||||||
Rat | Vas deferens | Inhibition | P2Y | α,β-MeATP | Suramin | ||
β,γ-MeATP | |||||||
2MeSATP | |||||||
Rat | Iris | Inhibition | P2Y | ATP | Reactive blue | Suramin | Fuder and Muth, 1993 |
α,β-MeATP | DIDS | ||||||
Mouse | Vas deferens | Inhibition | P2Y | Suramin | von Kugelgen et al., 1993 | ||
Reactive blue 2 | |||||||
Rabbit | Ear artery | Facilitation | P2 | ATP | Suramin | Ishii et al., 1993 | |
Rat | Iris | Inhibition | P2 | ATP | UTP | Fuder et al., 1992 | |
Rat | Vas deferens | Inhibition | P3 | 2-Chloroadenosine | 8-SPT | Forsyth et al., 1991 | |
ATP | α,β-MeATP | ||||||
β,γ-MeATP | |||||||
UTP | |||||||
Guinea pig | Ileum | Facilitation | P2X | α,β-MeATP | Sperlagh and Vizi, 1991 | ||
Rat | Caudal artery | Inhibition | P3 | 2-Chloroadenosine | α,β-MeATP | Shinozuka et al., 1990 | |
β,γ-MeATP | |||||||
Mouse | Vas deferens | Inhibition | P2Y | ATPγS | α,β-MeATP | von Kugelgen et al., 1989 | |
ATP | Uridine | ||||||
UTP | |||||||
Rat | Caudal artery | Inhibition | P3 | 2-Chloroadenosine | 8-SPT | Shinozuka et al., 1988 | |
β,γ-MeATP | |||||||
ATP | |||||||
Adenosine | |||||||
Rabbit | Ear artery | Facilitation | P2 | ATP | α,β-MeATP | Miyahara and Suzuki, 1987 | |
AMP-PNP2-i |
↵2-a β,γ-MeATP, β,γ-methylene ATP.
↵2-b DPCPX, 1,3-dipropyl-8-cyclopentylxanthine.
↵2-c 2MeSATP, 2-methylthio-ATP.
↵2-d PPADS, pyridoxalphosphate-6-azophenyl-2′,4′-disulfonic acid.
↵2-e α,β-MeATP, α,β-methylene ATP.
↵2-f TNP-ATP, 2′-o-(trinitrophenyl)-adenosine 5′-triphosphate.
↵2-g ATPγS, adenosine 5′[γ-thio]triphosphate.
↵2-h 8-SPT, 8-(p-sulfophenyl)-theophylline.
↵2-i AMP-PNP, adenosine 5′-[β,γ-imino]triphosphate.