Family | IUPHAR Receptor Code | Ligand | Official IUPHAR Nomenclature | Human Gene Symbol | Human Gene ID | Mouse Gene ID | Rat Gene ID |
---|---|---|---|---|---|---|---|
5-Hydroxytryptamine | 2.1:5HT:1:5HT1A: | 5-Hydroxytryptamine | 5-HT1A | HTR1A | 3350 | 15550 | 24473 |
5-Hydroxytryptamine | 2.1:5HT:2:5HT1B: | 5-Hydroxytryptamine | 5-HT1B | HTR1B | 3351 | 15551 | 25075 |
5-Hydroxytryptamine | 2.1:5HT:3:5HT1D: | 5-Hydroxytryptamine | 5-HT1D | HTR1D | 3352 | 15552 | 25323 |
5-Hydroxytryptamine | 2.1:5HT:4:5HT1E: | 5-Hydroxytryptamine | 5-HT1e | HTR1E | 3354 | ||
5-Hydroxytryptamine | 2.1:5HT:5:5HT1F: | 5-Hydroxytryptamine | 5-HT1F | HTR1F | 3355 | 15557 | 60448 |
5-Hydroxytryptamine | 2.1:5HT:6:5HT2A: | 5-Hydroxytryptamine | 5-HT2A | HTR2A | 3356 | 15558 | 29595 |
5-Hydroxytryptamine | 2.1:5HT:7:5HT2B: | 5-Hydroxytryptamine | 5-HT2B | HTR2B | 3357 | 15559 | 29581 |
5-Hydroxytryptamine | 2.1:5HT:8:5HT2C: | 5-Hydroxytryptamine | 5-HT2C | HTR2C | 3358 | 15560 | 25187 |
5-Hydroxytryptamine | 2.1:5HT:9:5HT4: | 5-Hydroxytryptamine | 5-HT4 | HTR4 | 3360 | 15562 | 25324 |
5-Hydroxytryptamine | 5-Hydroxytryptamine | 5-HT5A | HTR5A | 3361 | 15563 | 25689 | |
5-Hydroxytryptamine | 2.1:5HT:10:5HT6: | 5-Hydroxytryptamine | 5-HT6 | HTR6 | 3362 | 15565 | 64354 |
5-Hydroxytryptamine | 2.1:5HT:11:5HT7: | 5-Hydroxytryptamine | 5-HT7 | HTR7 | 3363 | 15566 | 65032 |
Acetylcholine (muscarinic) | 2.1:ACH:1:M1A: | Acetylcholine | M1 | CHRM1 | 1128 | 12669 | 25229 |
Acetylcholine (muscarinic) | 2.1:ACH:2:M2A: | Acetylcholine | M2 | CHRM2 | 1129 | 107850 | 81645 |
Acetylcholine (muscarinic) | 2.1:ACH:4:M2B: | Acetylcholine | M3 | CHRM4 | 1132 | 12672 | 25111 |
Acetylcholine (muscarinic) | 2.1:ACH:3:M1B: | Acetylcholine | M4 | CHRM3 | 1131 | 12671 | 24260 |
Acetylcholine (muscarinic) | 2.1:ACH:5:M1C: | Acetylcholine | M5 | CHRM5 | 1133 | 12673 | 53949 |
Adenosine | 2.1:ADO:1:A1: | Adenosine | A1 | ADORA1 | 134 | 11539 | 29290 |
Adenosine | 2.1:ADO:2:A2A: | Adenosine | A2A | ADORA2A | 135 | 11540 | 25369 |
Adenosine | 2.1:ADO:3:A2B: | Adenosine | A2B | ADORA2B | 136 | 11541 | 29316 |
Adenosine | 2.1:ADO:4:A3: | Adenosine | A3 | ADORA3 | 140 | 11542 | 25370 |
Adrenoceptors | 2.1:ADR:1:A1A: | Noradrenaline | α1A | ADRA1A | 148 | 11549 | 29412 |
Adrenoceptors | 2.1:ADR:2:A1B: | Adrenaline | α1B | ADRA1B | 147 | 11548 | 24173 |
Adrenoceptors | 2.1:ADR:3:A1D: | Adrenaline | α1D | ADRA1D | 146 | 11550 | 29413 |
Adrenoceptors | 2.1:ADR:4:A2A: | Adrenaline | α2A | ADRA2A | 150 | 11551 | 25083 |
Adrenoceptors | 2.1:ADR:5:A2B: | Adrenaline | α2B | ADRA2B | 151 | 11552 | 24174 |
Adrenoceptors | 2.1:ADR:6:A2C: | Adrenaline | α2c | ADRA2C | 152 | 11553 | 24175 |
Adrenoceptors | 2.1:ADR:7:B1: | Noradrenaline | β1 | ADRB1 | 153 | 11554 | 24925 |
Adrenoceptors | 2.1:ADR:8:B2: | Adrenaline | β2 | ADRB2 | 154 | 11555 | 24176 |
Adrenoceptors | 2.1:ADR:9:B3: | Adrenaline | β3 | ADRB3 | 155 | 11556 | 25645 |
Anaphylatoxin | Anaphylatoxin C5a, C5a des Arg74 | GPR77 | 27202 | 319430 | 445269 | ||
Anaphylatoxin | Anaphylatoxin C5a | C5R1 | 728 | 12273 | 113959 | ||
Anaphylatoxin | Anaphylatoxin C3a | C3AR1 | 719 | 12267 | 84007 | ||
Angiotensin | 2.1:ANG:1:AT1: | Angiotensin | AT1 | AGTR1 | 185 | 11607 | 81638 |
Angiotensin | 2.1:ANG:2:AT2: | Angiotensin | AT2 | AGTR2 | 186 | 11609 | 24182 |
Apelin | 2.1:APJ:1:APJ: | Apelin | AGTRL1 | 187 | 23796 | 83518 | |
Bombesin | 2.1:BB:1:BB1: | Neuromedin B | BB1 | NMBR | 4829 | 18101 | 25264 |
Bombesin | 2.1:BB:2:BB2: | Gastrin-releasing peptide | BB2 | GRPR | 2925 | 14829 | 24938 |
Bombesin | 2.1:BB:3:BB3: | BB3 | BRS3 | 680 | 12209 | 260319 | |
Bradykinin | 2.1:BK:1:B1: | Bradykinin | B1 | BDKRB1 | 623 | 12061 | 81509 |
Bradykinin | 2.1:BK:2:B2: | Bradykinin | B2 | BDKRB2 | 624 | 12062 | 25245 |
Cannabinoid | 2.1:CB:1:CB1: | Cannabinoid | CB1 | CNR1 | 1268 | 12801 | 25248 |
Cannabinoid | 2.1:CB:2:CB2: | Cannabinoid | CB2 | CNR2 | 1269 | 12802 | 57302 |
Chemokine | 2.1:CHK:1:CXC1: | CXCL8 | CXCR1 | IL8RA | 3577 | 227288 | 54258 |
Chemokine | 2.1:CHK:2:CXC2: | CXCL1—3, CXCL5—8 | CXCR2 | IL8RB | 3579 | 12765 | 29385 |
Chemokine | 2.1:CHK:3:CXC3: | CXCL9—11 | CXCR3 | CXCR3 | 2833 | 12766 | 84475 |
Chemokine | 2.1:CHK:4:CXC4: | CXCL12 | CXCR4 | CXCR4 | 7852 | 12767 | 60628 |
Chemokine | 2.1:CHK:5:CXC5: | CXCL13 | CXCR5 | BLR1 | 643 | 12145 | 29363 |
Chemokine | 2.1:CHK:6:CC1: | CCL3, CCL5, CCL7, CCL8, CCL13—16, CCL23 | CCR1 | CCR1 | 1230 | 12768 | 57301 |
Chemokine | 2.1:CHK:7:CC2: | CCL2, CCL7, CCL8, CCL13 | CCR2 | CCR2 | 1231 | 12772 | 60463 |
Chemokine | 2.1:CHK:8:CC3: | CCL11 (eotaxin); CCL5, CCL7, CCL8, CCL13, CCL15, CCL24, CCL26 | CCR3 | CCR3 | 1232 | 12771 | 117027 |
Chemokine | 2.1:CHK:9:CC4: | CCL17, CCL22 | CCR4 | CCR4 | 1233 | 12773 | 171054 |
Chemokine | 2.1:CHK:10:CC5: | CCL3, CCL4, CCL5, CCL8, CCL14 | CCR5 | CCR5 | 1234 | 12774 | 117029 |
Chemokine | 2.1:CHK:11:CC6: | CCL20 | CCR6 | CCR6 | 1235 | 12458 | |
Chemokine | 2.1:CHK:12:CC7: | CCL19, CCL21 | CCR7 | CCR7 | 1236 | 12775 | 287673 |
Chemokine | 2.1:CHK:13:CC8: | CCL1, CCL4, CCL17 | CCR8 | CCR8 | 1237 | 12776 | |
Chemokine | 2.1:CHK:14:CC9: | CCL25 | CCR9 | CCR9 | 10803 | 12769 | 282832 |
Chemokine | 2.1:CHK:15:CC10: | CCL26—28 | CCR10 | CCR10 | 2826 | 12777 | 363682 |
Chemokine | 2.1:CHK:17:CX3C1: | CX3CL1 | CX3CR1 | CX3CR1 | 1524 | 13051 | 171056 |
Chemokine | 2.1:CHK:18:XC1: | XCL1, XCL2 | XCR1 | XCR1 | 2829 | 23832 | 301086 |
Chemokine | 2.1:CHK:19:CXC6: | CXCL16 | CXCR6 | 10663 | 80901 | ||
Cholecystokinin | 2.1:CCK:1:CCK1: | Cholecystokinin | CCK1 | CCKAR | 886 | 12425 | 24889 |
Cholecystokinin | 2.1:CCK:2:CCK2: | Cholecystokinin, gastrin | CCK2 | CCKBR | 887 | 12426 | 25706 |
Dopamine | 2.1:DA:1:D1A: | Dopamine | D1 | DRD1 | 1812 | 13488 | 25678 |
Dopamine | 2.1:DA:2:D2A: | Dopamine | D2 | DRD2 | 1813 | 13489 | 24318 |
Dopamine | 2.1:DA:3:D2B: | Dopamine | D3 | DRD3 | 1814 | 13490 | 29238 |
Dopamine | 2.1:DA:4:D2C: | Dopamine | D4 | DRD4 | 1815 | 13491 | 25432 |
Dopamine | 2.1:DA:5:D1B: | Dopamine | D5 | DRD5 | 1816 | 13492 | 25195 |
Endothelin | 2.1:ET:1:ETA: | Endothelin 1, endothelin 2 | ETA | EDNRA | 1909 | 13617 | 24326 |
Endothelin | 2.1:ET:2:ETB: | Endothelins 1, 2 and 3 | ETB | EDNRB | 1910 | 13618 | 50672 |
Free fatty acid | 2.1:FFA:3:FFA3 | Acetate | GPR43 | 2867 | 233079 | 292794 | |
Free fatty acid | 2.1:FFA:2:FFA2 | Carboxylic acids | GPR41 | 2865 | 365228 | ||
Free fatty acid | GPR42a | 2866 | |||||
Free fatty acid | 2.1:FFA:1:FFA1 | Long chain carboxylic acids | GPR40 | 2864 | 233081 | 266607 | |
G protein-coupled bile acid | 2.1:BA:1:BA | Bile acids | GPBAR1 | 151306 | 227289 | ||
Galanin | 2.1:GAL:1:GAL1: | Galanin | GAL1 | GALR1 | 2587 | 14427 | 50577 |
Galanin | 2.1:GAL:2:GAL2: | Galanin | GAL2 | GALR2 | 8811 | 14428 | 29234 |
Galanin | 2.1:GAL:3:GAL3: | Galanin | GAL3 | GALR3 | 8484 | 14429 | 29235 |
Motilin | 2.1:MTLN:1:MTLN | Motilin | Motilin | MLNR | 2862 | ||
Ghrelin | 2.1:GRLN:1:GRLN | Ghrelin | Ghrelin | GHSR | 2693 | 208188 | 84022 |
Glycoprotein hormone | 2.1:GLYC:3:FSH: | Follicle-stimulating hormone | FSHR | 2492 | 14309 | 25449 | |
Glycoprotein hormone | 2.1:GLYC:2:LHCG: | Luteinizing hormone, chorionic gonadotropin | LHCGR | 3973 | 16867 | 25477 | |
Glycoprotein hormone | 2.1:GLYC:1:TSH: | Thyroid-stimulating hormone | TSHR | 7253 | 22095 | 25360 | |
GnRH | 2.1:GNRH:1:GNRH1: | Gonadotrophin-releasing hormone | GNRHR | 2798 | 14715 | 81668 | |
GnRH | Gonadotrophin-releasing hormone | GNRHR2 | 114814 | ||||
Histamine | 2.1:HIST:1:H1: | Histamine | H1 | HRH1 | 3269 | 15465 | 24448 |
Histamine | 2.1:HIST:2:H2: | Histamine | H2 | HRH2 | 3274 | 15466 | 25461 |
Histamine | 2.1:HIST:3:H3: | Histamine | H3 | HRH3 | 11255 | 99296 | 85268 |
Histamine | 2.1:HIST:4:H4: | Histamine | H4 | HRH4 | 59340 | 225192 | 170704 |
KiSS1-derived peptide | 2.1:KISS:1:KISS | KiSS-1 gene product | GPR54 | 84634 | 114229 | 78976 | |
Leukotriene and lipoxin | 2.1:LT:1:CLT1: | Leukotriene D4 | CysLT1 | CYSLTR1 | 10800 | 58861 | 114099 |
Leukotriene and lipoxin | 2.1:LT:2:CLT2: | Leukotriene C4 | CysLT2 | CYSLTR2 | 57105 | 70086 | 170926 |
Leukotriene and lipoxin | 2.1:LT:3:BLT1: | Leukotriene B4 | BLT1 | LTB4R | 1241 | 16995 | 59264 |
Leukotriene and lipoxin | 2.1:LT:4:BLT2: | Leukotriene B4 | BLT2 | LTB4R2 | 56413 | 57260 | 114098 |
Leukotriene and lipoxin | 2.1:LT:5:OXE: | 5-Oxo-6,8,11,14-eicosatetraenoic acid | OXE | OXER1 | 165140 | ||
Leukotriene and lipoxin | 2.1:LT:6:ALX: | Lipoxin Ab | ALX | FPRL1 | 2358 | 14294 | 171328 |
Lysophospholipid | 2.1:LPL:LPA1: | Lysophosphatidic acid | LPA1 | EDG2 | 1902 | 14745 | 116744 |
Lysophospholipid | 2.1:LPL:LPA2: | Lysophosphatidic acid | LPA2 | EDG4 | 9170 | 53978 | |
Lysophospholipid | 2.1:LPL:LPA3: | Lysophosphatidic acid | LPA3 | EDG7 | 23566 | 65086 | 66025 |
Lysophospholipid | 2.1:LPL:SIP1: | Sphingosine 1-phosphate | S1P1 | EDG1 | 1901 | 13609 | 29733 |
Lysophospholipid | 2.1:LPL:SIP2: | Sphingosine 1-phosphate | S1P2 | EDG5 | 9294 | 14739 | 29415 |
Lysophospholipid | 2.1:LPL:S1P3: | Sphingosine 1-phosphate | S1P3 | EDG3 | 1903 | 13610 | 29736 |
Lysophospholipid | 2.1:LPL:SIP4: | Sphingosine 1-phosphate | S1P4 | EDG6 | 8698 | 13611 | 314649 |
Lysophospholipid | 2.1:LPL:SIP5: | Sphingosine 1-phosphate | S1P5 | EDG8 | 53637 | 94226 | 60399 |
Melanin-concentrating hormone | 2.1:MCH:1:MCH1: | Melanin-concentrating hormone | MCH1 | GPR24 | 2847 | 207911 | 83567 |
Melanin-concentrating hormone | 2.1:MCH:2:MCH2: | Melanin-concentrating hormone | MCH2 | GPR145 | 84539 | ||
Melanocortin | 2.1:MC:1:MC1: | α-Melanocyte stimulating hormone | MC1 | MC1R | 4157 | 17199 | 292083 |
Melanocortin | 2.1:MC:2:MC2: | Adrenocorticotropic hormone | MC2 | MC2R | 4158 | 17200 | 282839 |
Melanocortin | 2.1:MC:3:MC3: | γ-Melanocyte stimulating hormone | MC3 | MC3R | 4159 | 17201 | 29310 |
Melanocortin | 2.1:MC:4:MC4: | β-Melanocyte stimulating hormone | MC4 | MC4R | 4160 | 17202 | 25635 |
Melanocortin | 2.1:MC:5:MC5: | α-Melanocyte stimulating hormone | MC5 | MC5R | 4161 | 17203 | 25726 |
Melatonin | 2.1:MLT:1:MT1: | Melatonin | [MT1] | MTNR1A | 4543 | 17773 | 114211 |
Melatonin | 2.1:MLT:1:MT2: | Melatonin | [MT2] | MTNR1B | 4544 | 244701 | 192646 |
Neuromedin U | 2.1:NMU:2:NMU2 | Neuromedin U | NMU2 | NMUR2 | 56923 | 216749 | 64042 |
Neuromedin U | 2.1:NMU:1:NMU1 | Neuromedin U | NMU1 | NMUR1 | 10316 | 14767 | 65276 |
Neuropeptide FF/neuropeptide AF | Neuropeptide FF | GPR147 | 64106 | 64107 | |||
Neuropeptide FF/neuropeptide AF | Neuropeptide FF | GPR74 | 10886 | 104443 | 78964 | ||
Neuropeptide S | Neuropeptide S | GPR154 | 387129 | 319239 | |||
Neuropeptide W/neuropeptide B | Neuropeptide W, neuropeptide B | GPR8 | 2832 | ||||
Neuropeptide W/neuropeptide B | Neuropeptide W, neuropeptide B | GPR7 | 2831 | 14769 | 297795 | ||
Neuropeptide Y | 2.1:NPY:1:Y1: | Neuropeptide Y | Y1 | NPY1R | 4886 | 18166 | 29358 |
Neuropeptide Y | 2.1:NPY:2:Y2: | Neuropeptide Y | Y2 | NPY2R | 4887 | 18167 | 66024 |
Neuropeptide Y | 2.1:NPY:3:Y4: | Pancreatic polypeptide | Y4 | PPYR1 | 5540 | 19065 | 29471 |
Neuropeptide Y | 2.1:NPY:4:Y5: | Neuropeptide Y | Y5 | NPY5R | 4889 | 18168 | 25340 |
Neurotensin | 2.1:NTSN:1:NTS1: | Neurotensin | NTS1 | NTSR1 | 4923 | 18216 | 366274 |
Neurotensin | 2.1:NTSN:2:NTS2: | Neurotensin | NTS2 | NTSR2 | 23620 | 18217 | 64636 |
N-Formylpeptide family | FPRL2 | 2359 | |||||
N-Formylpeptide family | N-Formyl-l-Met-l-Leu-l-Phe (fMLP) | FPR1 | 2357 | 14293 | |||
Nicotinic acid | GPR81 | 27198 | 243270 | ||||
Nicotinic acid | Nicotinic acid (low affinity) | GPR109B | 8843 | ||||
Nicotinic acid | Nicotinic acid (high affinity) | GPR109A | 338442 | 80885 | 353250 | ||
Opioid | 2.1:OP:2:DELTA: | β-Endorphin | δ | OPRD1 | 4985 | 18386 | 24613 |
Opioid | 2.1:OP:3:KAPPA: | Dynorphin A | κ | OPRK1 | 4986 | 18387 | 29335 |
Opioid | 2.1:OP:1:MU: | β-Endorphin | μ | OPRM1 | 4988 | 18390 | 25601 |
Opioid | 2.1:OP:4:NOCIC: | Nociceptin/orphanin FQ | NOP | OPRL1 | 4987 | 18389 | 29256 |
Opsin-like | OPN3 | 23596 | 13603 | ||||
Orexin (hypocretin) | Orexin A, orexin B | OX1 | HCRTR1 | 3061 | 230777 | 25593 | |
Orexin (hypocretin) | Orexin A, orexin B | OX2 | HCRTR2 | 3062 | 387285 | 25605 | |
P2Y | 2.1:NUCT:1:P2Y1: | ADP | P2Y1 | P2RY1 | 5028 | 18441 | 25265 |
P2Y | 2.1:NUCT:2:P2Y2: | UTP, ATP | P2Y2 | P2RY2 | 5029 | 18442 | 29597 |
P2Y | 2.1:NUCT:3:P2Y4: | UTP | P2Y4 | P2RY4 | 5030 | 57385 | 63843 |
P2Y | 2.1:NUCT:4:P2Y6: | UDP | P2Y6 | P2RY6 | 5031 | 233571 | 117264 |
P2Y | 2.1:NUCT:5:P2Y11: | ATP | P2Y11 | P2RY11 | 5032 | ||
P2Y | 2.1:NUCT:6:P2Y12: | ADP | [P2Y12] | P2RY12 | 64805 | 70839 | 64803 |
P2Y | 2.1:NUCT:7:P2Y13: | ADP | [P2Y13] | P2RY13 | 53829 | 74191 | 310444 |
P2Y | UDP-Glucose | P2RY14 | 9934 | 140795 | 171108 | ||
Peptide P518 | RF-Amide P518 gene productc | GPR103 | 84109 | 243407 | |||
Platelet-activating factor | 2.1:PAF:1:PAF | Platelet-activating factor | PAF | PTAFR | 5724 | 19204 | 58949 |
Prokineticin | 2.1:PROK:1:PK1 | Prokineticins 1 and 2 | PK1 | GPR73 | 10887 | 58182 | 192648 |
Prokineticin | 2.1:PROK:2:PK2 | Prokineticins 1 and 2 | PK2 | GPR73L1 | 128674 | 246313 | 192649 |
Prolactin-releasing peptide | 2.1:PRP:1:PRP | Prolactin-releasing peptide | PRP | GPR10 | 2834 | 226278 | 246075 |
Prostanoid | 2.1:PG:1:DP: | Prostaglandin D2 | DP | PTGDR | 5729 | 19214 | 63889 |
Prostanoid | 2.1:PG:2:EP1: | Prostaglandin E2 | EP1 | PTGER1 | 5731 | 19216 | 25637 |
Prostanoid | 2.1:PG:3:EP2: | Prostaglandin E2 | EP2 | PTGER2 | 5732 | 19217 | 81752 |
Prostanoid | 2.1:PG:4:EP3: | Prostaglandin E2 | EP3 | PTGER3 | 5733 | 19218 | 24929 |
Prostanoid | 2.1:PG:5:EP4: | Prostaglandin E2 | EP4 | PTGER4 | 5734 | 19219 | 84023 |
Prostanoid | 2.1:PG:6:FP: | Prostaglandin F2a | FP | PTGFR | 5737 | 19220 | 25652 |
Prostanoid | 2.1:PG:7:IP: | Prostacyclin | IP1 | PTGIR | 5739 | 19222 | 292661 |
Prostanoid | 2.1:PG:8:TP: | Thromboxane A2 | TP | TBXA2R | 6915 | 21390 | 24816 |
Prostanoid | 11-Dehydrothromboxane B2c | GPR44 | 11251 | 14764 | 29406 | ||
Protease-activated | 2.1:PAR:1:PAR1 | Thrombin | PAR1 | F2R | 2149 | 14062 | 25439 |
Protease-activated | 2:1:PAR:2:PAR2 | Serine proteases | PAR2 | F2RL1 | 2150 | 14063 | 116677 |
Protease-activated | 2.1:PAR:3:PAR3 | Thrombin | PAR3 | F2RL2 | 2151 | 14064 | 29636 |
Protease-activated | 2.1:PAR:4:PAR4 | Serine proteases | PAR4 | F2RL3 | 9002 | 14065 | 116498 |
Relaxin | Relaxin | LGR7 | 59350 | 381489 | |||
Relaxin | Relaxin | LGR8 | 122042 | 170458 | 171158 | ||
Relaxin | Relaxin-3 | RLN3R1 | 51289 | 239336 | 294807 | ||
Relaxin | INSL5, relaxin-3 | RLN3R2 | 339403 | 242093 | |||
Somatostatin | 2.1:SRIF:1:SRIF1A: | Somatostatin | sst2 | SSTR2 | 6752 | 20606 | 54305 |
Somatostatin | 2.1:SRIF:2:SRIF1B: | Somatostatin | sst5 | SSTR5 | 6755 | 20609 | 25354 |
Somatostatin | 2.1:SRIF:3:SRIF1C: | Somatostatin | sst3 | SSTR3 | 6753 | 20607 | 171044 |
Somatostatin | 2.1:SRIF:4:SRIF2A: | Somatostatin | sst1 | SSTR1 | 6751 | 20605 | 25033 |
Somatostatin | 2.1:SRIF:5:SRIF2B: | Somatostatin | sst4 | SSTR4 | 6754 | 20608 | 25555 |
SPC/LPC | (lyso)Phospholipid mediatorsd | GPR65 | 8477 | 14744 | 299242 | ||
SPC/LPC | (lyso)Phospholipid mediatorsd | GPR4 | 2828 | 319197 | 308408 | ||
SPC/LPC | (lyso)Phospholipid mediatorsd | GPR68 | 8111 | 238377 | |||
SPC/LPC | (lyso)Phospholipid mediatorsd | GPR132 | 29933 | 56696 | 314480 | ||
Tachykinin | 2.1:TAC:1:NK1: | Substance P | NK1 | TACR1 | 6869 | 21336 | 24807 |
Tachykinin | 2.1:TAC:2:NK2: | Neurokinin A | [NK2] | TACR2 | 6865 | 21337 | 25007 |
Tachykinin | 2.1:TAC:3:NK3: | Neurokinin B | NK3 | TACR3 | 6870 | 21338 | 24808 |
Trace Amine | β-Phenylethylamine, tyraminec | [TA1] | TRAR1 | 134864 | 111174 | 113914 | |
TRH | 2.1:TRH:1:TRH: | Thyrotropin-releasing hormone | TRH | TRHR | 7201 | 22045 | 25570 |
Urotensin | 2.1:UT:1:UT1: | Urotensin II | UT | UTS2R | 2837 | 217369 | 57305 |
Vasopressin/oxytocin | 2.1:OXY:1:OT: | Oxytocin | OT | OXTR | 5021 | 18430 | 25342 |
Vasopressin/oxytocin | 2.1:VASO:1:V1A: | Vasopressin | V1A | AVPR1A | 552 | 54140 | 25107 |
Vasopressin/oxytocin | 2.1:VASO:2:V2: | Vasopressin | V2 | AVPR2 | 554 | 12000 | 25108 |
Vasopressin/oxytocin | 2.1:VASO:3:V1B: | Vasopressin | V1B | AVPR1B | 553 | 26361 | 29462 |
OrphanA1 | Sphingosine 1-phosphatec | GPR3 | 2827 | 14748 | 266769 | ||
OrphanA1 | Sphingosine 1-phosphatec | GPR12 | 2835 | 14738 | 80840 | ||
OrphanA1 | Sphingosine 1-phosphatec | GPR6 | 2830 | 140741 | 83683 | ||
OrphanA2 | GPR52 | 9293 | |||||
OrphanA2 | GPR21 | 2844 | 338346 | ||||
OrphanA3 | GPR78 | 27201 | |||||
OrphanA3 | GPR26 | 2849 | 233919 | 192153 | |||
OrphanA4 | GPR37 | 2861 | 14763 | 117549 | |||
OrphanA4 | GPR37L1 | 9283 | 171469 | 252939 | |||
OrphanA6 | GPR63 | 81491 | 81006 | 297952 | |||
OrphanA6 | GPR45 | 11250 | 93690 | 301372 | |||
OrphanA7 | GPR83 | 10888 | 14608 | 140595 | |||
OrphanA9 | GRCAe | 27239 | 14788 | 362436 | |||
OrphanA9 | GPR153 | 387509 | 100129 | ||||
OrphanA12 | Lysophosphatidic acidc | GPR23 | 2846 | 78134 | 302378 | ||
OrphanA12 | P2RY5 | 10161 | 67168 | ||||
OrphanA13 | P2RY10 | 27334 | 78826 | 317219 | |||
OrphanA13 | GPR174 | 84636 | |||||
OrphanA14 | GPR142 | 350383 | 217302 | 303661 | |||
OrphanA14 | GPR139 | 124274 | 293545 | ||||
OrphanA15 | ADMR | 11318 | 11536 | 29307 | |||
OrphanA15 | CMKOR1 | 57007 | 12778 | 84348 | |||
OrphanLGR | LGR4 | 55366 | 107515 | 286994 | |||
OrphanLGR | LGR5 | 8549 | 14160 | 299802 | |||
OrphanLGR | LGR6 | 59352 | |||||
OrphanSREB | GPR85 | 54329 | 64450 | 64020 | |||
OrphanSREB | GPR27 | 2850 | 14761 | 65275 | |||
OrphanSREB | GPR173 | 54328 | 70771 | 64021 | |||
Orphan | Succinatec | SUCNR1 | 56670 | 84112 | 408199 | ||
Orphan | α-Ketoglutaratec | OXGR1 | 27199 | 239283 | 290493 | ||
Orphan (chemokine receptor-like) | CCRL2 | 9034 | 54199 | ||||
Orphan (Mas-related) | MAS1 | 4142 | 17171 | 25153 | |||
Orphan (Mas-related) | MAS1L | 116511 | |||||
Orphan (Mas-related) | β-Alaninec | MRGPRD | 116512 | ||||
Orphan (Mas-related) | MRGPRE | 116534 | |||||
Orphan (Mas-related) | MRGPRF | 116535 | |||||
Orphan (Mas-related) | MRGPRG | 386746 | |||||
Orphan (Mas-related) | BAM8—22c | MRGX1e | 259249 | 282547 | |||
Orphan (Mas-related) | Cortistatinc | MRGX2e | 117194 | ||||
Orphan (Mas-related) | MRGX3e | 117195 | |||||
Orphan (Mas-related) | MRGX4e | 117196 | |||||
Orphan (melatonin-like) | GPR50 | 9248 | 14765 | 117097 | |||
Orphan (P2Y-like) | GPR87 | 53836 | 84111 | ||||
Orphan (trace amine-like) | [TA3] | TRAR3f | 134860 | 319107 | |||
Orphan (trace amine-like) | [TA4] | TRAR4 | 319100 | 294124 | |||
Orphan (trace amine-like) | [TA5] | TRAR5 | 83551 | ||||
Orphan (trace amine-like) | PNRe | 9038 | 294123 | ||||
Orphan (trace amine-like) | GPR57g | 9288 | |||||
Orphan (trace amine-like) | GPR58 | 9287 | 294121 | ||||
Other orphan genes | RARRES2c | CMKLR1 | 1240 | 14747 | 60669 | ||
Other orphan genes | EBI2 | 1880 | 321019 | 306193 | |||
Other orphan genes | GPR160 | 26996 | 71862 | ||||
Other orphan genes | GPRe | 11245 | 117257 | ||||
Other orphan genes | GPR1 | 2825 | 241070 | 25457 | |||
Other orphan genes | GPR101 | 83550 | 317608 | ||||
Other orphan genes | GPR119 | 139760 | 236781 | ||||
Other orphan genes | GPR120 | 338557 | 107221 | 294075 | |||
Other orphan genes | GPR135 | 64582 | 314213 | ||||
Other orphan genes | OPN5 | 221391 | 353344 | 316259 | |||
Other orphan genes | GPR141 | 353345 | 353346 | 291179 | |||
Other orphan genes | GPR146 | 115330 | 80290 | ||||
Other orphan genes | GPR148 | 344561 | |||||
Other orphan genes | GPR149 | 344758 | 229357 | 192251 | |||
Other orphan genes | GPR15 | 2838 | 288181 | ||||
Other orphan genes | GPR150 | 285601 | 238725 | ||||
Other orphan genes | GPR152 | 390212 | 269053 | ||||
Other orphan genes | GPR161 | 23432 | 289180 | ||||
Other orphan genes | GPR17 | 2840 | |||||
Other orphan genes | GPR171 | 29909 | 229323 | ||||
Other orphan genes | GPR18 | 2841 | 110168 | 306191 | |||
Other orphan genes | GPR19 | 2842 | 14760 | 140664 | |||
Other orphan genes | GPR20 | 2843 | 239530 | 60667 | |||
Other orphan genes | GPR22 | 2845 | 73010 | ||||
Other orphan genes | GPR25 | 2848 | 363993 | ||||
Other orphan genes | GPR30 | 2852 | 76854 | 171104 | |||
Other orphan genes | GPR31 | 2853 | 107431 | 292310 | |||
Other orphan genes | GPR32 | 2854 | |||||
Other orphan genes | GPR33 | 2856 | 14762 | 299007 | |||
Other orphan genes | GPR34 | 2857 | 23890 | ||||
Other orphan genes | GPR35 | 2859 | 64095 | ||||
Other orphan genes | GPR39 | 2863 | 71111 | ||||
Other orphan genes | GPR55 | 9290 | |||||
Other orphan genes | GPR61 | 83873 | 229714 | 310780 | |||
Other orphan genes | GPR62 | 118442 | |||||
Other orphan genes | GPR75 | 10936 | 237716 | ||||
Other orphan genes | GPR79h | 27200 | |||||
Other orphan genes | GPR82 | 27197 | 319200 | ||||
Other orphan genes | GPR84 | 53831 | 80910 | 367000 | |||
Other orphan genes | GPR88 | 54112 | 64378 | 64443 | |||
Other orphan genes | GPR92 | 57121 | |||||
Other orphan genes | P2RY8 | 286530 | |||||
Other orphan genes | GPR151 | 134391 | 240239 | 307475 |
BAM8—22, 15 amino acid C-terminal fragment of bovine adrenal medulla peptide 22.
↵ a Very closely related to GPR41. May be a pseudogene
↵ b Under review by IUPHAR
↵ c Proposed ligand(s) supported by a single publication
↵ d Sphingosine-1-phosphate, lysophosphatidic acid, sphingosylphosphorylcholine, and phosphatidic acid
↵ e Interim gene symbol. The official symbol and name have not been established
↵ f A polymorphism introduces a stop codon in some individuals
↵ g May be a pseudogene
↵ h Probable pseudogene