Receptor | Recognized Agonist(s) | EC50 Range |
---|---|---|
FFA1 (GPR40 | Fatty acids (C6-C22) | Micromolar |
FFA2 (GPR43) | Fatty acids (C1-C6) | Micromolar to millimolar |
FFA3 (GPR41) | Fatty acids (C1-C6) | Micromolar to millimolar |
GPR84 | Fatty acids (C9-C14) | Micromolar |
GPR120 | Fatty acids (C14-C22) | Micromolar |
GPR3 | Sphingosine-1-phosphate? | |
GPR6 | Sphingosine-1-phosphate? | |
GPR12 | Sphingosylphosphorylcholine? | |
GPR18 | LPA | Nanomolar to micromolar |
Farnesyl pyrophosphate | Nanomolar to micromolar | |
NAGly | Nanomolar to micromolar | |
GPR23 | LPA? | |
GPR119 | OEA/OLDA | Low micromolar |
OEA, oleoyl ethanolamide; OLDA, N-oleoyl dopamine.