Dopamine receptor agonists and antagonists that have been used clinically
The table was compiled from information presented in articles cited in the text and from the references cited therein.
Drugs | Major Clinical Application |
---|---|
Dopamine agonists | |
Apomorphine | PD, erectile dysfunction |
Bromocriptine | PD, pituitary tumors, hyperprolactinemia, type 2 diabetes |
Cabergoline | Pituitary tumors, hyperprolactinemia |
Fenoldopam | Hypertension |
Pramipexole | PD, restless legs syndrome, bipolar disorder, depression |
Piribedil | PD |
Pergolide | PD |
Ropinirole | PD, restless legs syndrome |
Rotigotine | PD, bipolar disorder and depression |
Dopamine antagonists | |
Amisulpride | Schizophrenia, bipolar disorder, depression |
Aripiprazole | Schizophrenia, bipolar disorder, depression |
Benperidol | Schizophrenia |
Bromopride | Nausea, gastroparesis |
Chlorpromazine | Schizophrenia |
Clopenthixol | Schizophrenia |
Clozapine | Schizophrenia |
Domperidone | Nausea |
Droperidol | Schizophrenia, nausea |
Fluphenazine | Schizophrenia |
Flupentixol | Schizophrenia, depression |
Fluspirilene | Schizophrenia |
Haloperidol | Schizophrenia |
Quetiapine | Schizophrenia, bipolar disorder, depression |
Metoclopramide | Nausea, gastroparesis |
Olanzapine | Schizophrenia, bipolar disorder, depression |
Penfluridol | Schizophrenia |
Perazine | Schizophrenia |
Perphenazine | Schizophrenia |
Pimozide | Schizophrenia |
Prochlorperazine | Schizophrenia, nausea |
Promazine | Schizophrenia |
Risperidone | Schizophrenia, bipolar disorder |
Remoxipride | Schizophrenia |
Sertindole | Schizophrenia |
Sulpiride | Schizophrenia, depression |
Sultopride | Schizophrenia |
Thiethylperazine | Nausea |
Thiothixene | Schizophrenia |
Thioridazine | Schizophrenia |
Tiapride | Schizophrenia |
Trifluperidol | Schizophrenia |
Triflupromazine | Schizophrenia, nausea |
Trifluoperazine | Schizophrenia |
Ziprasidone | Schizophrenia, bipolar disorder, depression |