| nM | | |
Agonist | | | | |
BAM8–22 | 14 | | HEK293-Gαqi5 | Lembo et al., 2002 |
25 | | HEK293 | Burstein et al., 2006 |
40 | | HEK293 | Tatemoto et al., 2006 |
8–50 | | CHO | Kunapuli et al., 2006 |
150 | | HEK293 | Solinski et al., 2013 |
BAM1–22 | 16 | | HEK293-Gαqi5 | Lembo et al., 2002 |
800 | | HEK293 | Burstein et al., 2006 |
80 | | CHO-Gα16 | Shemesh et al., 2008 |
800 | | HEK293 | Malik et al., 2009 |
Chloroquine | 300,000 | | HEK293 | Liu et al., 2009 |
Benzimidazole derivates | 320 | | HEK293 | Malik et al., 2009 |
Antagonist | | | | |
Cyclic γ2-MSH6–12 derivates | | 12 | HEK293-Gαqi5 | Schmidt et al., 2009 |
Diaminopyrimidine derivates | | 14 | HEK293-Gαqi5 | Bayrakdarian et al., 2011 |
Azabicyclooctane derivates | | 100 | CHO | Kunapuli et al., 2006 |