TABLE 5

Ligand-binding affinities of SST2-selective ligands

SST1SST2SST3SST4SST5
L-779/976a27600.057293104260
BIM-23120b>10000.34412>1000213.5
DOTA-JR11c>10000.58>1000>1000>1000
  • a Data from Rohrer et al. (1998).

  • b Data from Gruszka et al. (2012).

  • c Data from Cescato et al. (2008).