TABLE 9

Ligand-binding affinities for approved and investigational SRIF ligands

SST1SST2SST3SST4SST5
Octreotidea>10000.44.4>10005.6
Lanreotideb21290.759818265.2
Pasireotidec9.311.5>1000.16
Veldoreotided>10003>10076
  • a Data from Reisine and Bell (1995), Patel (1999).

  • b Data from Shimon et al. (1997b), Zatelli et al. (2001).

  • c Data from Bruns et al. (2002).

  • d Data from Afargan et al. (2001).