TABLE 4

Bifunctional bronchodilator drugs and bifunctional bronchodilator/anti-inflammatory drugs

ClassSubgroupMolecules
Bifunctional bronchodilator drugsMABAsBatefenterol, AZD8871, LAS190792, CHF6366
Bifunctional bronchodilator/anti-inflammatory drugsPDE3–PDE4 inhibitorsEnsifentrine
PDE4–PDE5 inhibitorsLASSBio596
NO–ICSTPI 1020
NO–β2-AR agonistNCX 950
PDE4 inhibitor–β2-AR agonistGS-5759
PDE4 inhibitor–mAChR antagonistUCB-101333-3
Vasoactive intestinal peptide–pituitary AC-activating polypeptide type 2 receptorRO 50-24118